SCHEMBL8154102

SCHEMBL8154102

CC(C)(C)ON=O.[O-][N+](=S)c1ccc(-c2ccccc2)cc1Br

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 4/20 0.32
ABCC1 P33527 2/20 0.31
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
CRHBP P24387 2/20 0.30
CRHR2 Q13324 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4608252 0.82 CRHBP (0.42) ABCB1ABCC1CRHBPCRHR2
SCHEMBL30145522 0.70 CRHBP (0.53) ABCB1ABCC1CYP11B1CYP11B2CRHBP
SCHEMBL14928247 0.70 CRHBP (0.53) ABCB1ABCC1CYP11B1CYP11B2CRHBP
SCHEMBL4609299 0.67 MAPT (0.48) CRHBPCRHR2
SCHEMBL4608316 0.66 ABCB1 (0.44) ABCB1ABCC1
SCHEMBL8365480 0.62 ABCB1 (0.49) ABCB1ABCC1CRHBPCRHR2
SCHEMBL16997449 0.61 TDP1 (0.50) ABCB1ABCC1CYP11B1CYP11B2CRHBP
SCHEMBL2601600 0.61 CRHBP (0.58) ABCB1ABCC1CRHBPCRHR2
SCHEMBL9197991 0.61 AAK1 (0.60)
SCHEMBL14928233 0.61 MEN1 (0.51) ABCB1ABCC1CYP11B1CYP11B2CRHBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1059927-A1 CHEMICAL COMPOUNDS AND THEIR USE TO ELEVATE PYRUVATE DEHYDROGENASE ACTIVITY AstraZeneca AB (SE) 2000-12-20 EP disclosed
WO-1999044618-A1 CHEMICAL COMPOUNDS AND THEIR USE TO ELEVATE PYRUVATE DEHYDROGENASE ACTIVITY ASTRAZENECA AB (SE) 1999-09-10 WO disclosed