SCHEMBL8154173

SCHEMBL8154173

C=C(c1ccc(C#Cc2ccccc2)cc1)N1CCC(NC2CCC2)CC1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 8/20 0.48
MMP2 P08253 3/20 0.36
MMP9 P14780 3/20 0.36
EPHX1 P07099 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
CASP3 P42574 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
MMP12 P39900 1/20 0.36
PTGES O14684 1/20 0.36
EPHX2 P34913 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8161960 0.96 GRM5 (0.47) GRM5MMP2MMP9LMNAMMP12
SCHEMBL3643275 0.84 GRM5 (0.69) GRM5EPHX1MEN1LMNARAB9A
SCHEMBL8163323 0.82 GRM5 (0.69) GRM5MMP2MMP9KDM4EMEN1
SCHEMBL8168370 0.81 GRM5 (0.45) GRM5MMP2MMP9EPHX1KDM4E
SCHEMBL3641476 0.81 GRM5 (0.67) GRM5EPHX1KDM4EMEN1LMNA
SCHEMBL8154357 0.80 L3MBTL3 (0.52) GRM5
SCHEMBL8160754 0.80 L3MBTL3 (0.49) GRM5
SCHEMBL8161856 0.78 GRM5 (0.50) GRM5MMP2MMP9MMP12
SCHEMBL8162167 0.77 GRM5 (0.44) GRM5MMP2MMP9NPC1RAB9A
SCHEMBL8159305 0.76 GRM5 (0.48) GRM5MMP2MMP9KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008151184-A1 BENZAMIDE MGLUR5 POSITIVE ALLOSTERIC MODULATORS AND METHODS OF MAKING AND USING SAME VANDERBILT UNIVERSITY (US) 2008-12-11 WO disclosed