SCHEMBL8154259

SCHEMBL8154259

C=C(c1ccc(C#Cc2ccccc2)cc1)N1CCC(C)(O)CC1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRM3 Q14832 1/20 0.52
GRM5 P41594 11/20 0.46
CYP26A1 O43174 1/20 0.36
CYP3A4 P08684 1/20 0.36
RARA P10276 1/20 0.36
RARB P10826 1/20 0.36
RARG P13631 1/20 0.36
CRABP2 P29373 1/20 0.36
LMNA P02545 2/20 0.35
HTT P42858 1/20 0.35
MEN1 O00255 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8166489 0.87 GRM3 (0.51) GRM3GRM5
SCHEMBL8161987 0.86 GRM3 (0.46) GRM3GRM5
SCHEMBL8160780 0.86 GRM3 (0.46) GRM3GRM5
SCHEMBL8155708 0.85 GRM5 (0.44) GRM3GRM5CYP26A1CYP3A4RARA
SCHEMBL8168267 0.85 OPRM1 (0.46) GRM3GRM5RARARARBRARG
SCHEMBL8166622 0.84 CA12 (0.45) GRM5LMNAALDH1A1POLB
SCHEMBL3638549 0.83 GRM3 (0.74) GRM3GRM5LMNAHTTMEN1
SCHEMBL8159187 0.83 GRM5 (0.41) GRM3GRM5LMNAHTTALDH1A1
SCHEMBL8155823 0.83 GRM3 (0.47) GRM3GRM5CYP26A1CYP3A4RARA
SCHEMBL8162119 0.81 GRM5 (0.68) GRM5ALDH1A1POLBMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008151184-A1 BENZAMIDE MGLUR5 POSITIVE ALLOSTERIC MODULATORS AND METHODS OF MAKING AND USING SAME VANDERBILT UNIVERSITY (US) 2008-12-11 WO disclosed