SCHEMBL8155708

SCHEMBL8155708

C=C(c1ccc(C#Cc2ccccc2)cc1)N1CC(C)(O)C1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 13/20 0.44
GRM3 Q14832 1/20 0.39
APP P05067 1/20 0.36
CYP26A1 O43174 1/20 0.35
CYP3A4 P08684 1/20 0.35
RARA P10276 1/20 0.35
RARB P10826 1/20 0.35
RARG P13631 1/20 0.35
CRABP2 P29373 1/20 0.35
MMP2 P08253 1/20 0.35
MMP9 P14780 1/20 0.35
MMP12 P39900 1/20 0.35
MMP14 P50281 1/20 0.35
MMP15 P51511 1/20 0.35
MMP16 P51512 1/20 0.35
MMP26 Q9NRE1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8154259 0.85 GRM3 (0.52) GRM5GRM3CYP26A1CYP3A4RARA
SCHEMBL8164563 0.82 GRM5 (0.40) GRM5MMP2MMP9MMP12MMP14
SCHEMBL3640039 0.82 GRM5 (0.62) GRM5GRM3
SCHEMBL8162119 0.77 GRM5 (0.68) GRM5
SCHEMBL8168267 0.76 OPRM1 (0.46) GRM5GRM3RARARARBRARG
SCHEMBL8166622 0.75 CA12 (0.45) GRM5
SCHEMBL8166450 0.75 GRM5 (0.52) GRM5GRM3APPMMP2MMP9
SCHEMBL8171419 0.74 GRM5 (0.41) GRM5GRM3
SCHEMBL8160754 0.74 L3MBTL3 (0.49) GRM5
SCHEMBL8154357 0.74 L3MBTL3 (0.52) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008151184-A1 BENZAMIDE MGLUR5 POSITIVE ALLOSTERIC MODULATORS AND METHODS OF MAKING AND USING SAME VANDERBILT UNIVERSITY (US) 2008-12-11 WO disclosed