Phthalic Acid

Phthalic Acid

SCHEMBL8155

CCCC(=O)O.O=C(O)c1ccccc1C(=O)O

nearest known ligand 0.61

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.61
ALOX15 P16050 1/20 0.61
FFAR3 O14843 1/20 0.56
HDAC3 O15379 1/20 0.56
HDAC1 Q13547 1/20 0.56
HDAC2 Q92769 1/20 0.56
HDAC8 Q9BY41 1/20 0.56
HPGD P15428 3/20 0.52
HSD17B10 Q99714 1/20 0.52
KDM4E B2RXH2 2/20 0.50
MEN1 O00255 1/20 0.50
RECQL P46063 1/20 0.50
KMT2A Q03164 1/20 0.50
TDP1 Q9NUW8 1/20 0.48
ALOX5 P09917 1/20 0.48
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
AKR1C3 P42330 2/20 0.48
TSHR P16473 1/20 0.47
MYC P01106 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phthalic Acid SCHEMBL30717997 1.00 ALDH1A1 (0.61) ALDH1A1ALOX15FFAR3HDAC3HDAC1
Phthalic Acid SCHEMBL409472 0.96 ALDH1A1 (0.56) ALDH1A1ALOX15FFAR3HDAC3HDAC1
Salicylic Acid SCHEMBL28044508 0.88 ALDH1A1 (0.67) ALDH1A1ALOX15FFAR3HDAC3HDAC1
Toluic Acid SCHEMBL28104690 0.88 KMT2A (0.53) ALDH1A1ALOX15FFAR3HDAC3HDAC1
Butyric Acid SCHEMBL27907905 0.87 ALDH1A1 (0.53) ALDH1A1ALOX15FFAR3HDAC3HDAC1
Phthalic Acid SCHEMBL9132518 0.86 ALDH1A1 (0.74) ALDH1A1ALOX15HDAC8HPGDKDM4E
Phthalic Acid SCHEMBL22217134 0.86 ALDH1A1 (0.74) ALDH1A1ALOX15HDAC8HPGDHSD17B10
Phthalic Acid SCHEMBL1482851 0.86 ALDH1A1 (0.74) ALDH1A1ALOX15HDAC8HPGDKDM4E
Phthalic Acid SCHEMBL125858 0.86 ALDH1A1 (0.74) ALDH1A1ALOX15HDAC8HPGDHSD17B10
Phthalic Acid SCHEMBL6568928 0.86 AKR1B1 (0.61) ALDH1A1ALOX15HSD17B10KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2048 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024119044-A2 ADRULIPASE COMPOSITIONS First Wave BioPharma, Inc. (US) 2024-06-06 WO claimed
CN-118019524-A Dydrogesterone sustained release pharmaceutical composition 曼肯制药有限公司 2024-05-10 CN claimed
CN-114568676-B Composition for endowing food with tyrant flavor, and preparation method and application thereof 内蒙古伊利实业集团股份有限公司 2024-04-09 CN claimed
EP-3137060-B2 EXTENDED RELEASE SUSPENSION COMPOSITIONS SUN PHARMACEUTICAL IND LTD (IN) 2023-12-20 EP claimed
US-20230312606-A1 MCL-1 INHIBITOR FORMULATIONS AMGEN INC. (US) 2023-10-05 US claimed
WO-2023187599-A1 METHODS AND BIOAVAILABLE HIGHLY PERMEABLE COMPOUNDS FOR THE TREATMENT OF VIRAL DISEASES DIDENKO KIRILL (MX) 2023-10-05 WO claimed
CN-116437947-A Non-pig formulations and methods thereof 第一浪潮生物制药有限公司 2023-07-14 CN claimed
EP-4203922-A1 MCL-1 INHIBITOR FORMULATIONS Amgen Inc. (US) 2023-07-05 EP claimed
US-20230201164-A1 PHARMACEUTICAL COMPOSITION COMPRISING BENZIMIDAZOLE DERIVATIVE COMPOUND HK INNO.N CORPORATION (KR) 2023-06-29 US claimed
WO-2023114390-A2 LIPASE FORMULATIONS AND METHODS THEREOF First Wave BioPharma, Inc. (US) 2023-06-22 WO claimed
WO-1994003160-A1 PELLETISED PHARMACEUTICAL COMPOSITION F.H. FAULDING & CO. LIMITED (AU) 1994-02-17 WO claimed
EP-0241179-B1 PHARMACEUTICAL COMPOSITION FOR PERIODONTAL DISEASES ROHTO PHARMACEUTICAL CO., LTD. (JP) 1991-11-13 EP claimed
EP-0122815-B1 ENTERIC-SOLUBLE PREPARATIONS AND A PROCESS FOR THEIR PRODUCTION SANKYO COMPANY LIMITED (JP) 1989-10-25 EP claimed
EP-0241178-A1 Pharmaceutical composition for treating periodontal diseases ROHTO PHARMACEUTICAL CO., LTD. (JP) 1987-10-14 EP claimed
EP-0108504-B1 A PROCESS FOR COATING SOLID PHARMACEUTICAL PREPARATIONS AND COATED PREPARATIONS THUS OBTAINED SANKYO COMPANY LIMITED (JP) 1987-05-13 EP claimed
US-4661162-A MIXTURE OF POLYMER WITH POLYANIONIC POLYMER WHICH IS SOLUBLE AT LOW PH SANKYO COMPANY, LIMITED (JP) 1987-04-28 US claimed
US-4497847-A MONO AND DIESTERS OF GLYCEROL AND SATURATED CARBOXYLIC ACIDS AS PLASTICIZERS SANKYO COMPANY, LIMITED (JP) 1985-02-05 US claimed
EP-0122815-A1 Enteric-soluble preparations and a process for their production SANKYO COMPANY LIMITED (JP) 1984-10-24 EP claimed
EP-0108504-A1 A process for coating solid pharmaceutical preparations and coated preparations thus obtained SANKYO COMPANY LIMITED (JP) 1984-05-16 EP claimed
US-4134809-A GLYCIDYL ACRYLATES, ADHESIVE METAL COATINGS EASTMAN KODAK COMPANY (US) 1979-01-16 US claimed