SCHEMBL8155359

SCHEMBL8155359

Cc1cc2ccc(Br)cc2cc1C(N)=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.47
NCEH1 Q6PIU2 1/20 0.41
DHODH Q02127 2/20 0.41
MAPT P10636 5/20 0.41
KDM4E B2RXH2 3/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ALDH1A1 P00352 2/20 0.41
LCK P06239 1/20 0.41
MAOA P21397 1/20 0.40
CYP2A6 P11509 1/20 0.39
POLB P06746 1/20 0.39
MCL1 Q07820 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
LMNA P02545 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
F12 P00748 1/20 0.38
PARP1 P09874 1/20 0.38
NPC1 O15118 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8150190 1.00 DGAT1 (0.47) DGAT1NCEH1DHODHMAPTKDM4E
SCHEMBL8150396 0.82 NNMT (0.40) DGAT1KDM4EALDH1A1POLBL3MBTL1
SCHEMBL428805 0.80 DGAT1 (0.60) DGAT1MAPTKDM4EMEN1KMT2A
SCHEMBL1788262 0.80 DGAT1 (0.55) DGAT1MAPTKDM4EALDH1A1POLB
SCHEMBL31200433 0.80 DGAT1 (0.55) DGAT1MAPTKDM4EALDH1A1POLB
SCHEMBL8140936 0.80 IRAK4 (0.54) MAPTKDM4EMEN1KMT2AALDH1A1
SCHEMBL8153971 0.79 LCK (0.41) DGAT1MAPTKDM4EMEN1KMT2A
SCHEMBL8141517 0.79 KDM4E (0.50) MAPTKDM4EALDH1A1LCKCYP2A6
SCHEMBL8149236 0.79 KDM4E (0.50) MAPTKDM4EALDH1A1LCKCYP2A6
SCHEMBL8150193 0.79 LCK (0.41) DGAT1MAPTKDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040116399-A1 Inhibitors of factor Xa MILLENNIUM PHARMACEUTICALS, INC. 2004-06-17 US disclosed