SCHEMBL8156296

SCHEMBL8156296

Cc1cccc(-c2ccc3c(c2)CCNC3=O)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 10/20 1.00
PARP11 Q9NR21 10/20 1.00
GRM5 P41594 4/20 0.65
FYN P06241 1/20 0.61
CLK4 Q9HAZ1 1/20 0.61
DYRK1B Q9Y463 1/20 0.61
PARP1 P09874 2/20 0.56
PDPK1 O15530 1/20 0.50
PGR P06401 1/20 0.49
MAPKAPK2 P49137 2/20 0.48
GSK3B P49841 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16561672 0.86 PARP10 (0.76) PARP10PARP11GRM5CLK4PARP1
SCHEMBL13680532 0.85 CLK4 (0.78) PARP10PARP11GRM5FYNCLK4
SCHEMBL8155722 0.84 PARP11 (1.00) PARP10PARP11GRM5CLK4DYRK1B
SCHEMBL279903 0.82 PARP10 (1.00) PARP10PARP11GRM5PARP1PDPK1
SCHEMBL29978302 0.82 PARP10 (1.00) PARP10PARP11GRM5PARP1PDPK1
SCHEMBL8159245 0.82 PARP10 (1.00) PARP10PARP11GRM5PARP1PDPK1
SCHEMBL8154135 0.82 PARP10 (0.69) PARP10PARP11GRM5PARP1PDPK1
SCHEMBL20294385 0.82 PARP11 (0.72) PARP10PARP11GRM5PARP1PDPK1
SCHEMBL8154134 0.79 PARP11 (0.68) PARP10PARP11GRM5PARP1PDPK1
SCHEMBL23657097 0.79 PARP10 (0.65) PARP10PARP11GRM5PARP1PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008151184-A1 BENZAMIDE MGLUR5 POSITIVE ALLOSTERIC MODULATORS AND METHODS OF MAKING AND USING SAME VANDERBILT UNIVERSITY (US) 2008-12-11 WO disclosed