SCHEMBL8156328

SCHEMBL8156328

COc1ccc(-c2ccccc2)c(Cl)c1C1CCCN(C)C1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.48
HTR2C P28335 2/20 0.48
DRD2 P14416 1/20 0.48
KCNH2 Q12809 1/20 0.48
HTR1A P08908 1/20 0.43
HTR1D P28221 1/20 0.43
HTR1B P28222 1/20 0.43
HTR1E P28566 1/20 0.43
HTR7 P34969 1/20 0.43
HTR2B P41595 1/20 0.43
HTR3A P46098 1/20 0.43
HTR5A P47898 1/20 0.43
CHRNB2 P17787 1/20 0.42
CHRNB4 P30926 1/20 0.42
CHRNA3 P32297 1/20 0.42
CHRNA4 P43681 1/20 0.42
PDE3A Q14432 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CD274 Q9NZQ7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8137489 0.74 HTR2A (0.54) HTR2AHTR2CDRD2KCNH2
SCHEMBL12852526 0.71 HTR2A (0.56) HTR2AHTR2CDRD2MEN1KMT2A
SCHEMBL28740554 0.71 BRD4 (0.52) HTR2AHTR2CDRD2KCNH2CHRNB2
SCHEMBL11893151 0.67 DRD2 (0.65) HTR2AHTR2CDRD2KCNH2CHRNB2
SCHEMBL2077235 0.67 DRD2 (0.65) HTR2AHTR2CDRD2KCNH2CHRNB2
SCHEMBL13006443 0.67 DRD2 (0.65) HTR2AHTR2CDRD2KCNH2CHRNB2
Hydrochloric Acid SCHEMBL11627075 0.66 SLC6A2 (0.54) HTR2AHTR2CDRD2KCNH2HTR1A
SCHEMBL2277992 0.66 HTR2C (0.48) HTR2AHTR2CDRD2HTR1AHTR1D
SCHEMBL25722721 0.65 HTR2A (0.59) HTR2AHTR1AHTR7HTR2B
SCHEMBL8525408 0.65 HTR2A (1.00) HTR2AHTR2CDRD2KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1037876-A1 BIPHENYL DERIVATIVES AS PHARMACEUTICALS Novartis AG (CH) 2000-09-27 EP disclosed
WO-1999023073-A1 BIPHENYL DERIVATIVES AS PHARMACEUTICALS NOVARTIS AG (CH) 1999-05-14 WO disclosed