SCHEMBL8157768

SCHEMBL8157768

CC(O)OCCN1CCN(Cc2ccc(-c3cc4nccc(Nc5ccc6[nH]ccc6c5)c4s3)cc2)CC1

nearest known ligand 0.71

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
EGFR P00533 19/20 0.71
FLT1 P17948 19/20 0.71
PRKCQ Q04759 1/20 0.50
PRKCD Q05655 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8160355 0.90 FLT1 (0.67) EGFRFLT1PRKCQPRKCD
SCHEMBL7127760 0.88 EGFR (0.73) EGFRFLT1PRKCQPRKCD
SCHEMBL7126230 0.88 EGFR (0.79) EGFRFLT1PRKCQPRKCD
SCHEMBL7668263 0.85 EGFR (0.79) EGFRFLT1
SCHEMBL7127750 0.84 EGFR (0.76) EGFRFLT1PRKCQPRKCD
SCHEMBL7119457 0.83 EGFR (1.00) EGFRFLT1PRKCQPRKCD
SCHEMBL7126184 0.83 EGFR (0.78) EGFRFLT1PRKCQPRKCD
SCHEMBL7127685 0.80 EGFR (1.00) EGFRFLT1
SCHEMBL7127504 0.79 EGFR (0.72) EGFRFLT1PRKCQPRKCD
SCHEMBL7127001 0.79 EGFR (0.77) EGFRFLT1PRKCQPRKCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1028964-A1 THIENOPYRIMIDINE AND THIENOPYRIDINE DERIVATIVES USEFUL AS ANTICANCER AGENTS Pfizer Products Inc. (US) 2000-08-23 EP claimed
WO-1999024440-A1 THIENOPYRIMIDINE AND THIENOPYRIDINE DERIVATIVES USEFUL AS ANTICANCER AGENTS PFIZER PRODUCTS INC. (US) 1999-05-20 WO claimed
EP-1028964-A1 THIENOPYRIMIDINE AND THIENOPYRIDINE DERIVATIVES USEFUL AS ANTICANCER AGENTS Pfizer Products Inc. (US) 2000-08-23 EP disclosed
WO-1999024440-A1 THIENOPYRIMIDINE AND THIENOPYRIDINE DERIVATIVES USEFUL AS ANTICANCER AGENTS PFIZER PRODUCTS INC. (US) 1999-05-20 WO disclosed