SCHEMBL8166298

SCHEMBL8166298

CC(C)(C)N(NC(=O)c1ccccn1)C(=O)c1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.68
CYP3A4 P08684 2/20 0.59
CYP2C9 P11712 2/20 0.59
KMT2A Q03164 2/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
MEN1 O00255 1/20 0.49
LMNA P02545 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
MAPT P10636 1/20 0.49
CYP2C19 P33261 1/20 0.49
HTT P42858 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
RECQL P46063 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9426147 0.91 POLB (0.56) POLBCYP3A4CYP2C9KMT2ASMN1; SMN2
SCHEMBL8173935 0.90 POLB (0.55) POLBCYP3A4CYP2C9KMT2ASMN1; SMN2
SCHEMBL8173237 0.89 POLB (0.68) POLBCYP3A4CYP2C9KMT2A
SCHEMBL9425963 0.87 ABCB1 (0.64) POLBCYP3A4CYP2C9KMT2AMEN1
SCHEMBL9815842 0.87 HPGD (0.68) POLBCYP3A4SMN1; SMN2
SCHEMBL9425270 0.87 ABCB1 (0.64) POLBCYP3A4CYP2C9CYP2C19HTT
SCHEMBL9815875 0.86 POLB (0.72) POLBCYP3A4CYP2C9SMN1; SMN2RECQL
SCHEMBL8178669 0.85 POLB (0.63) POLBCYP3A4CYP2C9SMN1; SMN2RECQL
SCHEMBL8173402 0.85 MEN1 (0.55) POLBCYP3A4CYP2C9KMT2ASMN1; SMN2
SCHEMBL9815808 0.84 TLR7 (0.64) POLBCYP3A4CYP2C9KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5354762-A Insecticides ROHM AND HAAS COMPANY (US) 1994-10-11 US claimed
US-6013836-A PARTICULARLY ACTIVE AGAINST MOTHS AND BEETLES AND THEIR INSECT GROWTH REGULATING ACTIVITY WITHOUT ADVERSE IMPACT ON BENEFICIAL INSECTS; CROPS; FORESTRY ROHM AND HAAS COMPANY (US) 2000-01-11 US disclosed
US-5424333-A Anthelmintic N'-substituted-N,N'-disubstitutedhydrazines ROHM AND HAAS COMPANY (US) 1995-06-13 US disclosed
US-5354762-A Insecticides ROHM AND HAAS COMPANY (US) 1994-10-11 US disclosed
EP-0361645-B1 ORGANIC HYDRAZINE DERIVATIVES FOR PHARMACEUTICAL USE ROHM AND HAAS COMPANY (US) 1993-09-29 EP disclosed
US-5117057-A Insecticidal N' substituted-N-N'-disubstituted-hydrazines ROHM AND HAAS COMPANY (US) 1992-05-26 US disclosed
EP-0253468-B1 SIX-MEMBERED HETEROCYCLIC DERIVATIVES OF N'SUBSTITUTED-N,N'-DIACYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1991-11-06 EP disclosed
EP-0361645-A2 Organic hydrazine derivatives for pharmaceutical use ROHM AND HAAS COMPANY (US) 1990-04-04 EP disclosed
EP-0253468-A2 Six-membered heterocyclic derivatives of N'substituted-N,N'-diacylhydrazines ROHM AND HAAS COMPANY (US) 1988-01-20 EP disclosed