SCHEMBL8173237

SCHEMBL8173237

CC(C)(C)N(NC(=O)c1ccccc1)C(=O)c1ccccn1

nearest known ligand 0.68

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.68
CYP3A4 P08684 1/20 0.63
CYP2C9 P11712 1/20 0.63
KMT2A Q03164 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9815800 0.91 POLB (0.56) POLBCYP3A4CYP2C9KMT2A
SCHEMBL9511093 0.90 AGTR1 (0.55) POLBCYP3A4CYP2C9KMT2A
SCHEMBL8166298 0.89 POLB (0.68) POLBCYP3A4CYP2C9KMT2A
SCHEMBL9425189 0.87 HPGD (0.68) POLBCYP3A4CYP2C9
SCHEMBL9815864 0.87 ABCB1 (0.60) POLBCYP3A4CYP2C9
SCHEMBL9426130 0.86 POLB (0.72) POLBCYP3A4CYP2C9
SCHEMBL9425567 0.85 POLB (0.63) POLBCYP3A4CYP2C9
SCHEMBL9425890 0.84 TLR7 (0.64) POLBCYP3A4CYP2C9KMT2A
SCHEMBL9509589 0.84 MEN1 (0.57) POLBCYP3A4CYP2C9KMT2A
SCHEMBL9815862 0.84 POLB (0.65) POLBCYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6013836-A PARTICULARLY ACTIVE AGAINST MOTHS AND BEETLES AND THEIR INSECT GROWTH REGULATING ACTIVITY WITHOUT ADVERSE IMPACT ON BENEFICIAL INSECTS; CROPS; FORESTRY ROHM AND HAAS COMPANY (US) 2000-01-11 US disclosed
US-5424333-A Anthelmintic N'-substituted-N,N'-disubstitutedhydrazines ROHM AND HAAS COMPANY (US) 1995-06-13 US disclosed
US-5354762-A Insecticides ROHM AND HAAS COMPANY (US) 1994-10-11 US disclosed
EP-0361645-B1 ORGANIC HYDRAZINE DERIVATIVES FOR PHARMACEUTICAL USE ROHM AND HAAS COMPANY (US) 1993-09-29 EP disclosed
US-5117057-A Insecticidal N' substituted-N-N'-disubstituted-hydrazines ROHM AND HAAS COMPANY (US) 1992-05-26 US disclosed
EP-0253468-B1 SIX-MEMBERED HETEROCYCLIC DERIVATIVES OF N'SUBSTITUTED-N,N'-DIACYLHYDRAZINES ROHM AND HAAS COMPANY (US) 1991-11-06 EP disclosed
EP-0361645-A2 Organic hydrazine derivatives for pharmaceutical use ROHM AND HAAS COMPANY (US) 1990-04-04 EP disclosed
EP-0253468-A2 Six-membered heterocyclic derivatives of N'substituted-N,N'-diacylhydrazines ROHM AND HAAS COMPANY (US) 1988-01-20 EP disclosed