SCHEMBL8166369

SCHEMBL8166369

Cn1cc(C2=C(c3cn(CCCCCO)c4ccccc34)C(=O)NC2=O)c2ccccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 3/20 0.75
CAMK2D Q13557 1/20 0.75
GSK3B P49841 2/20 0.72
PRKCA P17252 2/20 0.72
PRKACA P17612 1/20 0.72
PRKACG P22612 1/20 0.72
PRKACB P22694 1/20 0.72
CCNE2 O96020 2/20 0.67
CDK4 P11802 2/20 0.67
CCND1 P24385 2/20 0.67
CCNE1 P24864 2/20 0.67
CDK2 P24941 2/20 0.67
MEN1 O00255 1/20 0.67
CASK O14936 1/20 0.67
CCNT1 O60563 1/20 0.67
RPS6KA5 O75582 1/20 0.67
CCNK O75909 1/20 0.67
STK10 O94804 1/20 0.67
PRKD3 O94806 1/20 0.67
TP53 P04637 1/20 0.67

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3150613 0.99 PIM1 (0.77) PIM1CAMK2DGSK3BPRKCAPRKACA
SCHEMBL3139598 0.95 GSK3B (0.78) PIM1CAMK2DGSK3BPRKCAPRKACA
SCHEMBL8161322 0.90 CCNE2 (0.74) PIM1CAMK2DGSK3BPRKCAPRKACA
SCHEMBL7873644 0.89 PRKACA (0.80) PIM1CAMK2DGSK3BPRKCAPRKACA
SCHEMBL8154114 0.88 CAMK2D (0.91) PIM1CAMK2DGSK3BPRKCAPRKACA
SCHEMBL8161268 0.86 CCNT1 (0.75) PIM1CAMK2DGSK3BPRKCAPRKACA
SCHEMBL8167286 0.86 PIM1 (0.76) PIM1CAMK2DGSK3BPRKCAPRKACA
Hydrochloric Acid SCHEMBL8160489 0.86 CAMK2D (0.91) PIM1CAMK2DGSK3BPRKCAPRKACA
SCHEMBL1942352 0.86 CAMK2D (1.00) PIM1CAMK2DPRKCAPRKACAPRKACG
SCHEMBL8161666 0.86 PIM1 (0.78) PIM1CAMK2DGSK3BPRKCAPRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE36736-E Substituted pyrroles HOFFMAN-LA ROCHE INC. (US) 2000-06-13 US disclosed
EP-0328026-B1 SUBSTITUTED PYRROLES F. HOFFMANN-LA ROCHE AG (CH) 1993-04-28 EP disclosed
US-5057614-A Antiinflammatory, immunology, bronchodilator agents, cardiovascular disorders HOFFMANN-LA ROCHE INC. (US) 1991-10-15 US disclosed
EP-0328026-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1989-08-16 EP disclosed