SCHEMBL8167454

SCHEMBL8167454

O=C1NC(=O)C(c2cn(CCCO)c3ccccc23)=C1c1ccccc1[N+](=O)[O-]

nearest known ligand 0.70

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 9/20 0.70
QPCT Q16769 6/20 0.70
CDK4 P11802 1/20 0.64
PRKACA P17612 1/20 0.64
PRKACG P22612 1/20 0.64
PRKACB P22694 1/20 0.64
CCND1 P24385 1/20 0.64
PRKCB P05771 1/20 0.61
PRKCA P17252 1/20 0.61
PRKCE Q02156 1/20 0.61
KDR P35968 1/20 0.58
FLT3 P36888 1/20 0.58
CAMK2D Q13557 1/20 0.57
IDH1 O75874 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7873644 0.88 PRKACA (0.80) GSK3BCDK4PRKACAPRKACGPRKACB
SCHEMBL8160483 0.85 GSK3B (0.65) GSK3BQPCTPRKACAPRKACGPRKACB
SCHEMBL13166904 0.84 CAMK2D (0.78) GSK3BQPCTCDK4PRKACAPRKACG
SCHEMBL8154930 0.83 GSK3B (0.68) GSK3BQPCTPRKACAPRKACGPRKACB
SCHEMBL1250687 0.82 GSK3B (0.72) GSK3BCDK4PRKACAPRKACGPRKACB
SCHEMBL30319781 0.82 GSK3B (0.72) GSK3BCDK4PRKACAPRKACGPRKACB
SCHEMBL3139598 0.82 GSK3B (0.78) GSK3BCDK4PRKACAPRKACGPRKACB
SCHEMBL5682666 0.81 GSK3B (0.62) GSK3BCDK4PRKACAPRKACGPRKACB
SCHEMBL5682520 0.81 GSK3B (0.62) GSK3BCDK4PRKACAPRKACGPRKACB
SCHEMBL30319769 0.81 GSK3B (0.62) GSK3BCDK4PRKACAPRKACGPRKACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE36736-E Substituted pyrroles HOFFMAN-LA ROCHE INC. (US) 2000-06-13 US disclosed
EP-0328026-B1 SUBSTITUTED PYRROLES F. HOFFMANN-LA ROCHE AG (CH) 1993-04-28 EP disclosed
US-5057614-A Antiinflammatory, immunology, bronchodilator agents, cardiovascular disorders HOFFMANN-LA ROCHE INC. (US) 1991-10-15 US disclosed
EP-0328026-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1989-08-16 EP disclosed