SCHEMBL8167493

SCHEMBL8167493

Cc1cccc(C2=C(c3cn(C)c4ccccc34)C(=O)OC2=O)c1

nearest known ligand 0.72

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 3/20 0.54
PRKCA P17252 2/20 0.54
CCNE2 O96020 1/20 0.51
CDK4 P11802 1/20 0.51
CCND1 P24385 1/20 0.51
CCNE1 P24864 1/20 0.51
CDK2 P24941 1/20 0.51
CCNT1 O60563 1/20 0.50
CDK9 P50750 1/20 0.50
CAMK2D Q13557 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8154180 0.84 GSK3B (0.76) GSK3BPRKCACCNE2CDK4CCND1
SCHEMBL4419603 0.82 GSK3B (0.49) GSK3BPRKCACCNE2CDK4CCND1
SCHEMBL8160875 0.79 CCNT1 (0.56) GSK3BPRKCACCNE2CDK4CCND1
SCHEMBL6581528 0.79 GSK3B (0.62) GSK3BPRKCACCNE2CDK4CCND1
SCHEMBL8161267 0.79 CDK2 (0.56) GSK3BPRKCACCNE2CDK4CCND1
SCHEMBL8162060 0.78 CDK2 (0.56) GSK3BPRKCACCNE2CDK4CCND1
SCHEMBL8154478 0.77 CDK2 (0.51) GSK3BPRKCACCNE2CDK4CCND1
SCHEMBL9667604 0.77 MAPT (0.49)
SCHEMBL8161370 0.76 CCNT1 (0.56) GSK3BCCNE2CDK4CCND1CCNE1
SCHEMBL8161741 0.76 PRKCA (0.56) GSK3BPRKCACCNE2CDK4CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE36736-E Substituted pyrroles HOFFMAN-LA ROCHE INC. (US) 2000-06-13 US disclosed
EP-0328026-B1 SUBSTITUTED PYRROLES F. HOFFMANN-LA ROCHE AG (CH) 1993-04-28 EP disclosed
US-5057614-A Antiinflammatory, immunology, bronchodilator agents, cardiovascular disorders HOFFMANN-LA ROCHE INC. (US) 1991-10-15 US disclosed
EP-0328026-A1 Substituted pyrroles F. HOFFMANN-LA ROCHE AG (CH) 1989-08-16 EP disclosed