SCHEMBL8170273

SCHEMBL8170273

CC1=Cc2c(cccc2-c2ccc3ccccc3c2)C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSTP1 P09211 1/20 0.43
HDAC4 P56524 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
MET P08581 1/20 0.39
DHFR P00374 1/20 0.39
BACE1 P56817 2/20 0.38
ACHE P22303 1/20 0.38
HSD17B1 P14061 1/20 0.38
HSD17B2 P37059 1/20 0.38
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
CYP2A6 P11509 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
AKT1 P31749 1/20 0.36
ESR2 Q92731 2/20 0.36
ESR1 P03372 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4469441 0.84 GSTP1 (0.40) GSTP1HDAC4HDAC2HDAC8SLC6A2
SCHEMBL26606289 0.83 NR1H2 (0.32) ALDH1A1HPGDKDM4E
SCHEMBL1827132 0.80 PDCD1 (0.39) CYP2A6ALDH1A1HPGDTSHRHSD17B10
SCHEMBL30229874 0.80 PDCD1 (0.39) CYP2A6ALDH1A1HPGDTSHRHSD17B10
SCHEMBL7863648 0.78 PDCD1 (0.38) CYP2A6ALDH1A1HPGDTSHRHSD17B10
Lithium SCHEMBL6324236 0.78 PDCD1 (0.38) CYP2A6ALDH1A1HPGDTSHRHSD17B10
SCHEMBL27185392 0.78 PDCD1 (0.38) CYP2A6ALDH1A1HPGDTSHRHSD17B10
SCHEMBL7643421 0.78 PDCD1 (0.38) CYP2A6ALDH1A1HPGDTSHRHSD17B10
SCHEMBL6324232 0.78 PDCD1 (0.38) CYP2A6ALDH1A1HPGDTSHRHSD17B10
SCHEMBL6330045 0.78 HTR1A (0.34) CYP2A6ALDH1A1CYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968158-A1 METHOD OF PREPARING SUBSTITUTED INDANONES, THE SUBSTITUTED INDANONES AND METALLOCENES PREPARED THEREFROM Basell Polyolefine GmbH (DE) 2000-01-05 EP disclosed
WO-1998040331-A1 PREPARATION OF PREPARING SUBSTITUTED INDANONES TARGOR GMBH (DE) 1998-09-17 WO disclosed