SCHEMBL8170686

SCHEMBL8170686

N=C(N)c1ccc(S(=O)(=O)NCc2ccccc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.65
PRMT1 Q99873 1/20 0.62
TMPRSS6 Q8IU80 7/20 0.61
CA12 O43570 2/20 0.60
CA9 Q16790 2/20 0.60
CYP1A2 P05177 1/20 0.60
CYP3A4 P08684 1/20 0.60
ATM Q13315 1/20 0.60
L3MBTL1 Q9Y468 1/20 0.60
CA1 P00915 1/20 0.59
CA2 P00918 1/20 0.59
ALDH1A1 P00352 3/20 0.56
F2 P00734 4/20 0.55
CYP19A1 P11511 1/20 0.54
PLAU P00749 1/20 0.53
HPN P05981 1/20 0.53
LMNA P02545 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
POLB P06746 2/20 0.52
KDM4E B2RXH2 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5449745 0.86 PRMT1 (0.68) KEAP1PRMT1CA12CA9CYP1A2
SCHEMBL15555895 0.83 TMPRSS6 (0.55) KEAP1TMPRSS6CA12CA9CA1
SCHEMBL4168948 0.82 KEAP1 (0.61) KEAP1PRMT1CA12CA9CYP1A2
SCHEMBL7972526 0.82 PRSS1 (0.58) PRMT1TMPRSS6F2PLAULMNA
SCHEMBL7972038 0.81 PRSS1 (0.59) PRMT1ALDH1A1F2PLAULMNA
SCHEMBL7986040 0.81 TMPRSS2 (0.59) PRMT1TMPRSS6ALDH1A1F2PLAU
SCHEMBL12348122 0.80 TMPRSS6 (0.58) TMPRSS6CA12CA9CYP3A4CA1
SCHEMBL28727051 0.80 CYP19A1 (0.81) KEAP1PRMT1CA12CA9CYP1A2
SCHEMBL407414 0.80 KEAP1 (1.00) KEAP1PRMT1CA12CA9CYP1A2
SCHEMBL7989750 0.80 PRMT1 (0.60) PRMT1ALDH1A1F2PLAULMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6114328-A ANTICOAGULANTS; BLOOD DISORDERS DUPONT PHARMACEUTICALS COMPANY (US) 2000-09-05 US disclosed
US-5849736-A Isoxazoline and isoxazole fibrinogen receptor antagonists THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-12-15 US disclosed
EP-0730590-A1 NOVEL ISOXAZOLINE AND ISOXAZOLE FIBRINOGEN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-09-11 EP disclosed