SCHEMBL8175997

SCHEMBL8175997

O=C1C(=Cc2ccc(-c3ccccc3[N+](=O)[O-])o2)SC(=S)N1c1cccc(O)c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K5 Q99683 1/20 0.66
HTRA2 O43464 2/20 0.58
INSR P06213 1/20 0.52
IGF1R P08069 1/20 0.52
MAPT P10636 4/20 0.52
MAPK1 P28482 2/20 0.52
TDP1 Q9NUW8 2/20 0.52
GSK3A P49840 1/20 0.51
GSK3B P49841 1/20 0.51
CDK2 P24941 1/20 0.51
PTPN12 Q05209 1/20 0.51
PTPN22 Q9Y2R2 1/20 0.51
HPGD P15428 2/20 0.49
LMNA P02545 1/20 0.49
GAA P10253 1/20 0.49
HTT P42858 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
PIK3CA P42336 1/20 0.49
PIK3CG P48736 1/20 0.49
BRAF P15056 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6279044 0.90 HTRA2 (0.71) MAP3K5HTRA2INSRIGF1RMAPT
SCHEMBL3897920 0.90 HTRA2 (0.71) MAP3K5HTRA2INSRIGF1RMAPT
SCHEMBL3897914 0.90 HTRA2 (0.71) MAP3K5HTRA2INSRIGF1RMAPT
SCHEMBL3892418 0.84 HTRA2 (0.61) HTRA2INSRIGF1RMAPTMAPK1
SCHEMBL3892423 0.84 HTRA2 (0.61) HTRA2INSRIGF1RMAPTMAPK1
SCHEMBL7168872 0.84 PTPN12 (0.72) HTRA2INSRIGF1RMAPTMAPK1
SCHEMBL6784929 0.84 PTPN12 (0.72) HTRA2INSRIGF1RMAPTMAPK1
SCHEMBL3900012 0.80 HTRA2 (0.55) HTRA2INSRIGF1RMAPTMAPK1
SCHEMBL3900015 0.80 HTRA2 (0.55) HTRA2INSRIGF1RMAPTMAPK1
SCHEMBL3894596 0.80 MAPT (0.65) MAP3K5HTRA2INSRIGF1RMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000032598-A9 METHODS AND COMPOSITIONS FOR TREATING INFLAMMATORY DISEASES UTILIZING INHIBITORS OF TUMOR NECROSIS FACTOR ACTIVITY STRUCTURAL BIOINFORMATICS INC (US) 2000-11-30 WO claimed
WO-2000032598-A1 METHODS AND COMPOSITIONS FOR TREATING INFLAMMATORY DISEASES UTILIZING INHIBITORS OF TUMOR NECROSIS FACTOR ACTIVITY STRUCTURAL BIOINFORMATICS INC. (US) 2000-06-08 WO claimed