SCHEMBL8176115

SCHEMBL8176115

N=C(N)c1cc[c]c(Nc2cccc3ccccc23)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLAU P00749 6/20 0.48
F2 P00734 4/20 0.48
PLG P00747 4/20 0.48
KLK1 P06870 3/20 0.48
PRSS1 P07477 3/20 0.48
PLAT P00750 2/20 0.48
SIRT2 Q8IXJ6 1/20 0.46
SIRT1 Q96EB6 1/20 0.46
SIRT3 Q9NTG7 1/20 0.46
KDM4E B2RXH2 1/20 0.43
GAA P10253 1/20 0.43
ALDH1A1 P00352 3/20 0.41
TP53 P04637 2/20 0.41
CDC25B P30305 2/20 0.41
TSHR P16473 2/20 0.41
HSD17B10 Q99714 2/20 0.41
CYP3A4 P08684 1/20 0.41
HPGD P15428 1/20 0.41
ALOX15 P16050 1/20 0.41
ATM Q13315 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8174776 0.78 PLAU (0.44) PLAUF2PLGKLK1PRSS1
SCHEMBL9630060 0.74 HSD17B10 (0.53) KDM4EGAAALDH1A1TP53CDC25B
SCHEMBL8169486 0.70 PRSS1 (0.39) PLAUF2PLGPRSS1ALDH1A1
SCHEMBL8169762 0.69 PRSS1 (0.46) PLAUF2PRSS1KLKB1BLM
SCHEMBL8170639 0.67 PLAU (0.38) PLAUF2PLGKLK1PRSS1
SCHEMBL8170185 0.67 PLAU (0.38) PLAUF2PLGKLK1PRSS1
SCHEMBL49213 0.67 HSD17B10 (0.74) KDM4EGAAALDH1A1TP53CDC25B
Ammonia Solution, Strong SCHEMBL11586421 0.65 HSD17B10 (0.71) KDM4EGAAALDH1A1TP53CDC25B
SCHEMBL8500339 0.65 HSD17B10 (0.71) KDM4EGAAALDH1A1TP53CDC25B
SCHEMBL1921580 0.65 HSD17B10 (0.71) KDM4EGAAALDH1A1TP53CDC25B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6114328-A ANTICOAGULANTS; BLOOD DISORDERS DUPONT PHARMACEUTICALS COMPANY (US) 2000-09-05 US disclosed
US-5849736-A Isoxazoline and isoxazole fibrinogen receptor antagonists THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-12-15 US disclosed
EP-0730590-A1 NOVEL ISOXAZOLINE AND ISOXAZOLE FIBRINOGEN RECEPTOR ANTAGONISTS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-09-11 EP disclosed