SCHEMBL8178461

SCHEMBL8178461

Cc1sc2nc(C3CCC(C(=O)O)CC3)nc(NCCc3ccccc3)c2c1C

nearest known ligand 0.62

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.62
LMNA P02545 2/20 0.56
MAPT P10636 1/20 0.56
ALOX15 P16050 1/20 0.56
HTT P42858 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
KDM4E B2RXH2 1/20 0.45
MAPK1 P28482 1/20 0.45
MAOB P27338 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8180123 0.91 ALDH1A1 (0.51) ALDH1A1LMNAMAPTALOX15
SCHEMBL8183118 0.90 ALDH1A1 (0.59) ALDH1A1LMNAMAPTALOX15HTT
Bicarbonate SCHEMBL7016458 0.89 ALDH1A1 (0.60) ALDH1A1LMNAMAPTALOX15HTT
SCHEMBL8178383 0.86 ALDH1A1 (0.51) ALDH1A1LMNAMAPTALOX15HTT
SCHEMBL8180824 0.86 ALDH1A1 (0.51) ALDH1A1LMNAMAPTALOX15HTT
SCHEMBL8170169 0.85 ALDH1A1 (0.44) ALDH1A1LMNAMAPTALOX15HTT
SCHEMBL8179115 0.83 ALDH1A1 (0.42) ALDH1A1SMN1; SMN2KDM4E
SCHEMBL8184348 0.82 HTT (0.49) ALDH1A1LMNAMAPTHTTSMN1; SMN2
SCHEMBL8181994 0.82 ALDH1A1 (0.52) ALDH1A1LMNAMAPTALOX15HTT
SCHEMBL8180882 0.81 PDE10A (0.53) ALDH1A1LMNAMAPTALOX15HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6130223-A Thienopyrimidine with phosphodiesterase V inhibiting effect MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-10-10 US disclosed