SCHEMBL8178656

SCHEMBL8178656

Cc1ccc(Oc2cccc(C3C4=C(CC(C)(C)CC4=O)NC4=C3C(=O)CC(C)(C)C4)c2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.59
KDM4E B2RXH2 9/20 0.59
HPGD P15428 7/20 0.59
GAA P10253 5/20 0.59
GSK3B P49841 5/20 0.56
GSK3A P49840 3/20 0.56
MAPT P10636 4/20 0.53
LMNA P02545 4/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
L3MBTL1 Q9Y468 2/20 0.53
NPC1 O15118 1/20 0.51
AURKA O14965 2/20 0.49
AURKB Q96GD4 2/20 0.49
INCENP Q9NQS7 2/20 0.49
HSD17B10 Q99714 3/20 0.48
MAPK1 P28482 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
GLA P06280 1/20 0.47
TSHR P16473 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8179019 0.92 KDM4E (0.59) ALDH1A1KDM4EHPGDGAAGSK3B
SCHEMBL8186789 0.91 KDM4E (0.64) ALDH1A1KDM4EHPGDGAAGSK3B
SCHEMBL8187896 0.90 ALDH1A1 (0.55) ALDH1A1KDM4EHPGDGAAGSK3B
SCHEMBL8194355 0.88 KDM4E (0.55) ALDH1A1KDM4EHPGDGAAGSK3B
SCHEMBL8186808 0.85 ALDH1A1 (0.55) ALDH1A1KDM4EHPGDGAAGSK3B
SCHEMBL8188863 0.83 KDM4E (0.58) ALDH1A1KDM4EHPGDGAAGSK3B
SCHEMBL7814828 0.83 GSK3B (0.69) ALDH1A1KDM4EHPGDGAAGSK3B
SCHEMBL7815046 0.80 KMT2A (0.70) ALDH1A1KDM4EHPGDGAAGSK3B
SCHEMBL8189185 0.79 KDM4E (0.51) ALDH1A1KDM4EHPGDGAAGSK3B
SCHEMBL2746217 0.78 L3MBTL1 (0.69) ALDH1A1KDM4EHPGDGAAGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6162918-A Xanthene and acridine derivatives HOFFMANN-LA ROCHE INC. (US) 2000-12-19 US disclosed
US-5969139-A INHIBITORS OF HERPES SIMPLEX VIRUS THYMIDINE KINASE HOFFMANN-LA ROCHE INC. (US) 1999-10-19 US disclosed
EP-0823426-A1 Xanthene and acridine derivatives and their use F. HOFFMANN-LA ROCHE AG (CH) 1998-02-11 EP disclosed