SCHEMBL8181737

SCHEMBL8181737

CC(I)(I)c1ccc2c(c1)OCO2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.45
ATM Q13315 1/20 0.43
SLC6A2 P23975 2/20 0.41
SLC6A3 Q01959 2/20 0.41
PGR P06401 1/20 0.41
AR P10275 1/20 0.41
GABRA1 P14867 1/20 0.41
MAOA P21397 1/20 0.41
PDE4A P27815 1/20 0.41
KDR P35968 1/20 0.41
GABRB2 P47870 1/20 0.41
ALDH1A1 P00352 4/20 0.41
HSD17B10 Q99714 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
MAPK9 P45984 2/20 0.41
MAPK1 P28482 1/20 0.40
TRPV1 Q8NER1 1/20 0.40
TAAR1 Q96RJ0 3/20 0.40
SLC6A4 P31645 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8284590 0.88 CYP3A4 (0.45) CYP3A4ATMSLC6A2SLC6A3PGR
SCHEMBL30567467 0.83 ALDH1A1 (0.52) CYP3A4ATMSLC6A2SLC6A3PGR
SCHEMBL85405 0.83 ALDH1A1 (0.52) CYP3A4ATMSLC6A2SLC6A3PGR
SCHEMBL14349288 0.80 CYP3A4 (0.45) CYP3A4ATMSLC6A2SLC6A3PGR
SCHEMBL20222611 0.80 CYP3A4 (0.45) CYP3A4ATMSLC6A2SLC6A3PGR
SCHEMBL933157 0.80 CYP3A4 (0.50) CYP3A4ATMSLC6A2SLC6A3PGR
SCHEMBL22338921 0.80 CYP3A4 (0.45) CYP3A4ATMSLC6A2SLC6A3PGR
SCHEMBL5288474 0.80 CYP3A4 (0.45) CYP3A4ATMSLC6A2SLC6A3PGR
Hydrochloric Acid SCHEMBL12614854 0.78 CYP3A4 (0.44) CYP3A4ATMSLC6A2SLC6A3PGR
SCHEMBL1744766 0.77 ALDH1A1 (0.52) CYP3A4ATMSLC6A2SLC6A3PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008077557-A1 8-ETHINYLXANTHINE DERIVATIVES AS SELECTIVE A2A RECEPTOR ANTAGONISTS SCHWARZ PHARMA AG (DE) 2008-07-03 WO disclosed