SCHEMBL8181971

SCHEMBL8181971

Cn1cc(-c2cn(COCC[Si](C)(C)C)c3ncccc23)cn1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 3/20 0.46
DGAT1 O75907 1/20 0.39
MAPT P10636 1/20 0.38
EGFR P00533 1/20 0.37
IGF1R P08069 1/20 0.37
SRC P12931 1/20 0.37
FLT4 P35916 1/20 0.37
KDR P35968 1/20 0.37
FLT3 P36888 1/20 0.37
EPHB4 P54760 1/20 0.37
TEK Q02763 1/20 0.37
GSK3B P49841 4/20 0.37
AURKA O14965 1/20 0.36
AURKB Q96GD4 1/20 0.36
INCENP Q9NQS7 1/20 0.36
TPX2 Q9ULW0 1/20 0.36
DYRK1A Q13627 1/20 0.35
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
PRKCB P05771 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31298196 0.83 DGAT1 (0.34) BRD4DGAT1MAPTEGFRIGF1R
SCHEMBL18789133 0.83 MKNK1 (0.42) BRD4DGAT1MAPTEGFRIGF1R
SCHEMBL31298152 0.82 KDR (0.37) BRD4DGAT1EGFRIGF1RSRC
SCHEMBL19832096 0.82 KDR (0.37) BRD4DGAT1EGFRIGF1RSRC
SCHEMBL8472530 0.82 DGAT1 (0.39) BRD4DGAT1EGFRIGF1RSRC
SCHEMBL19832083 0.82 JAK2 (0.40) BRD4DGAT1EGFRIGF1RSRC
SCHEMBL8470002 0.81 DGAT1 (0.36) BRD4DGAT1EGFRIGF1RSRC
SCHEMBL2753800 0.81 DGAT1 (0.41) BRD4DGAT1EGFRIGF1RSRC
SCHEMBL3347313 0.81 DGAT1 (0.36) BRD4DGAT1EGFRIGF1RSRC
SCHEMBL3355528 0.81 KDR (0.41) BRD4DGAT1EGFRIGF1RSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008095944-A1 7-AZAINDOLE DERIVATIVES AND THEIR USE IN THE INHIBITION OF C-JUN N-TERMINAL KINASE EISAI R&D MANAGEMENT CO. LTD. (JP) 2008-08-14 WO disclosed