SCHEMBL8470002

SCHEMBL8470002

Bc1cnc2c(c1)c(-c1cnn(C)c1)cn2COCC[Si](C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 6/20 0.36
BRD4 O60885 5/20 0.35
CREBBP Q92793 1/20 0.33
LRRK2 Q5S007 1/20 0.33
EGFR P00533 1/20 0.32
IGF1R P08069 1/20 0.32
SRC P12931 1/20 0.32
FLT4 P35916 1/20 0.32
KDR P35968 1/20 0.32
FLT3 P36888 1/20 0.32
EPHB4 P54760 1/20 0.32
TEK Q02763 1/20 0.32
AURKA O14965 2/20 0.31
AURKB Q96GD4 2/20 0.31
INCENP Q9NQS7 2/20 0.31
TPX2 Q9ULW0 2/20 0.31
ALOX5AP P20292 1/20 0.31
FEN1 P39748 1/20 0.31
MAP4K4 O95819 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8472530 0.88 DGAT1 (0.39) DGAT1BRD4CREBBPLRRK2EGFR
SCHEMBL2753800 0.87 DGAT1 (0.41) DGAT1BRD4CREBBPLRRK2EGFR
SCHEMBL3347313 0.87 DGAT1 (0.36) DGAT1BRD4CREBBPLRRK2EGFR
SCHEMBL3346630 0.85 BRD4 (0.37) DGAT1BRD4CREBBPLRRK2SRC
SCHEMBL13539153 0.85 DGAT1 (0.35) DGAT1BRD4CREBBPLRRK2EGFR
SCHEMBL3349611 0.84 BRD4 (0.36) DGAT1BRD4CREBBPLRRK2EGFR
SCHEMBL3352910 0.83 CYP19A1 (0.35) DGAT1BRD4CREBBP
SCHEMBL3353967 0.83 MET (0.40) DGAT1BRD4CREBBPLRRK2EGFR
SCHEMBL8445038 0.83 CHUK (0.37) DGAT1BRD4CREBBPEGFRIGF1R
SCHEMBL3352871 0.83 DGAT1 (0.36) DGAT1BRD4CREBBPLRRK2KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1749829-B1 JNK inhibitors EISAI R&D MAN CO LTD (JP) 2010-11-03 EP disclosed