SCHEMBL8184282

SCHEMBL8184282

COc1ccc(CNc2nc(C3CCC(C(=O)O)CC3)nc3sc(C)c(C)c23)cc1OC

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.48
LMNA P02545 2/20 0.46
MAPT P10636 1/20 0.46
ALOX15 P16050 1/20 0.46
GAA P10253 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
ACHE P22303 5/20 0.40
APP P05067 3/20 0.40
BCHE P06276 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
POLB P06746 2/20 0.39
HSP90AA1 P07900 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HTT P42858 1/20 0.39
CHRM4 P08173 1/20 0.39
NPC1 O15118 1/20 0.38
PKM P14618 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8179501 0.93 ALDH1A1 (0.46) ALDH1A1LMNAMAPTALOX15PDE10A
SCHEMBL8176737 0.92 ALDH1A1 (0.39) ALDH1A1LMNAMAPTALOX15ACHE
Bicarbonate SCHEMBL7017197 0.90 ALDH1A1 (0.47) ALDH1A1LMNAMAPTALOX15GAA
SCHEMBL8179863 0.86 ESR1 (0.42) ALDH1A1LMNAMAPTACHEAPP
SCHEMBL8179485 0.86 ALDH1A1 (0.49) ALDH1A1LMNAMAPTALOX15GAA
SCHEMBL8184358 0.86 PDE5A (0.45)
SCHEMBL8171487 0.86 MAPT (0.46) ALDH1A1LMNAMAPTGAAACHE
SCHEMBL8183118 0.85 ALDH1A1 (0.59) ALDH1A1LMNAMAPTALOX15GAA
SCHEMBL8178313 0.85 ACHE (0.44) ACHEAPPBCHEMEN1KMT2A
SCHEMBL8181994 0.85 ALDH1A1 (0.52) ALDH1A1LMNAMAPTALOX15GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6130223-A Thienopyrimidine with phosphodiesterase V inhibiting effect MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-10-10 US disclosed