SCHEMBL8190341

SCHEMBL8190341

CCCOc1cccc2c1CCN(C)C2

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.56
ADRA2A P08913 2/20 0.55
ADRA2B P18089 2/20 0.55
ADRA2C P18825 2/20 0.55
ACACB O00763 1/20 0.49
S1PR5 Q9H228 1/20 0.48
PRMT5 O14744 1/20 0.47
MAOA P21397 2/20 0.46
MAOB P27338 2/20 0.46
DRD2 P14416 1/20 0.44
DRD1 P21728 1/20 0.44
DRD5 P21918 1/20 0.44
DRD3 P35462 1/20 0.44
KDM4E B2RXH2 1/20 0.43
MAPT P10636 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
ABHD6 Q9BV23 1/20 0.41
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8190334 0.93 HRH3 (0.58) HRH3ADRA2AADRA2BADRA2CACACB
SCHEMBL8185348 0.90 S1PR5 (0.60) HRH3ADRA2AADRA2BADRA2CACACB
SCHEMBL8187016 0.88 HRH3 (0.56) HRH3ADRA2AADRA2BADRA2CS1PR5
SCHEMBL8187058 0.88 ADRA2A (0.57) HRH3ADRA2AADRA2BADRA2CACACB
Ammonia Solution, Strong SCHEMBL8185454 0.87 ADRA2A (0.56) HRH3ADRA2AADRA2BADRA2CACACB
SCHEMBL10571355 0.86 HRH3 (0.54) HRH3ADRA2AADRA2BADRA2CS1PR5
SCHEMBL11742426 0.86 HRH3 (0.64) HRH3ADRA2AADRA2BADRA2CACACB
SCHEMBL8192754 0.85 ADRA2A (0.51) HRH3ADRA2AADRA2BADRA2CS1PR5
SCHEMBL8190422 0.83 HRH3 (0.52) HRH3ADRA2AADRA2BADRA2CS1PR5
SCHEMBL8176552 0.81 S1PR5 (0.60) HRH3ADRA2AADRA2BADRA2CS1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6096752-A Method for the preparation of tertiary amines, a compound useful therefor and alpha-2-receptor active tetrahydroisoquinoline derivatives HEINONEN PETRI (FI) 2000-08-01 US disclosed
US-5912342-A SYNTHESIS OF COMBINATORIAL LIBRARIES BY COMPUTER CONTROLLED ROBOT HEINONEN PETRI (FI) 1999-06-15 US disclosed
EP-0910562-A2 A METHOD FOR THE PREPARATION OF TERTIARY AMINES, A COMPOUND USEFUL THEREFOR AND ALPHA-2-RECEPTOR ACTIVE TETRAHYDROISOQUINOLINE DERIVATIVES Oy Juvantia Pharma Ltd (FI) 1999-04-28 EP disclosed
WO-1998051672-A2 A METHOD FOR THE PREPARATION OF TERTIARY AMINES, A COMPOUND USEFUL THEREFOR AND ALPHA-2-RECEPTOR ACTIVE TETRAHYDROISOQUINOLINE DERIVATIVES OY JUVANTIA PHARMA LTD. (FI) 1998-11-19 WO disclosed