SCHEMBL8185463

SCHEMBL8185463

C[C@H](CO)COc1cccc2c1CN(C)CC2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 2/20 0.49
ADRA2B P18089 2/20 0.49
ADRA2C P18825 2/20 0.49
PRMT5 O14744 2/20 0.48
WDR77 Q9BQA1 1/20 0.48
DRD2 P14416 2/20 0.46
DRD1 P21728 2/20 0.46
DRD5 P21918 2/20 0.46
DRD3 P35462 2/20 0.46
HRH3 Q9Y5N1 1/20 0.43
TSHR P16473 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MAOA P21397 2/20 0.41
MAOB P27338 2/20 0.41
CYP2D6 P10635 1/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8185466 1.00 ADRA2A (0.49) ADRA2AADRA2BADRA2CPRMT5WDR77
SCHEMBL8189815 0.90 ADRA2A (0.49) ADRA2AADRA2BADRA2CPRMT5WDR77
SCHEMBL8189808 0.90 ADRA2A (0.49) ADRA2AADRA2BADRA2CPRMT5WDR77
SCHEMBL8187016 0.77 HRH3 (0.56) ADRA2AADRA2BADRA2CPRMT5WDR77
SCHEMBL25907679 0.76 DRD1 (0.54) ADRA2AADRA2BADRA2CPRMT5WDR77
SCHEMBL8187259 0.76 HRH3 (0.58) ADRA2AADRA2BADRA2CPRMT5WDR77
SCHEMBL8184418 0.75 CHRNA7 (0.61) ADRA2AADRA2BADRA2CPRMT5WDR77
SCHEMBL8187075 0.75 DRD2 (0.52) ADRA2AADRA2BADRA2CPRMT5WDR77
SCHEMBL5568684 0.74 DRD1 (0.77) ADRA2AADRA2BADRA2CDRD2DRD1
SCHEMBL8192779 0.74 HRH3 (0.53) ADRA2AADRA2BADRA2CPRMT5WDR77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6096752-A Method for the preparation of tertiary amines, a compound useful therefor and alpha-2-receptor active tetrahydroisoquinoline derivatives HEINONEN PETRI (FI) 2000-08-01 US disclosed
US-5912342-A SYNTHESIS OF COMBINATORIAL LIBRARIES BY COMPUTER CONTROLLED ROBOT HEINONEN PETRI (FI) 1999-06-15 US disclosed
EP-0910562-A2 A METHOD FOR THE PREPARATION OF TERTIARY AMINES, A COMPOUND USEFUL THEREFOR AND ALPHA-2-RECEPTOR ACTIVE TETRAHYDROISOQUINOLINE DERIVATIVES Oy Juvantia Pharma Ltd (FI) 1999-04-28 EP disclosed
WO-1998051672-A2 A METHOD FOR THE PREPARATION OF TERTIARY AMINES, A COMPOUND USEFUL THEREFOR AND ALPHA-2-RECEPTOR ACTIVE TETRAHYDROISOQUINOLINE DERIVATIVES OY JUVANTIA PHARMA LTD. (FI) 1998-11-19 WO disclosed