SCHEMBL8186402

SCHEMBL8186402

NC1=N[C@@H](Cc2ccccc2)CSc2ccsc21

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.44
NOS2 P35228 13/20 0.41
NOS3 P29474 9/20 0.41
NOS1 P29475 5/20 0.40
HDAC3 O15379 1/20 0.38
NCOR1 O75376 1/20 0.38
HDAC2 Q92769 1/20 0.38
NPC1 O15118 1/20 0.33
MAPT P10636 1/20 0.33
STAT3 P40763 1/20 0.33
HTT P42858 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8215252 0.84 TAAR1 (0.50) TAAR1NOS2NOS3NOS1
SCHEMBL8194863 0.80 NOS2 (0.47) NOS2NOS3NOS1
SCHEMBL8193587 0.80 NOS2 (0.47) NOS2NOS3NOS1
SCHEMBL8193125 0.78 NOS2 (0.58) NOS2NOS3NOS1
SCHEMBL8186361 0.76 NOS2 (0.61) TAAR1NOS2NOS3NOS1NPC1
SCHEMBL8197854 0.76 NOS2 (0.54) NOS2NOS3NOS1
SCHEMBL6191572 0.75 TAAR1 (0.51) TAAR1NOS2NOS3NOS1HDAC3
SCHEMBL6994968 0.75 TAAR1 (0.51) TAAR1NOS2NOS3NOS1HDAC3
Hydrochloric Acid SCHEMBL6752220 0.73 TAAR1 (0.50) TAAR1NOS2NOS3NOS1HDAC3
SCHEMBL8216232 0.73 TAAR1 (0.39) TAAR1NOS2NOS3NOS1HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000064904-A1 5,7-BICYCLIC AMIDINE DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS ASTRAZENECA AB (SE) 2000-11-02 WO claimed
WO-2000064904-A1 5,7-BICYCLIC AMIDINE DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS ASTRAZENECA AB (SE) 2000-11-02 WO disclosed