SCHEMBL8189740

SCHEMBL8189740

CCOP(=O)(OCC)c1csc(C(=O)O)c1C

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
POLB P06746 4/20 0.38
GPR35 Q9HC97 7/20 0.35
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.32
GSK3B P49841 1/20 0.32
KDM4E B2RXH2 1/20 0.32
PKM P14618 1/20 0.32
MAPK1 P28482 1/20 0.31
CASP1 P29466 1/20 0.31
CASP7 P55210 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3879287 0.69 TSHR (0.47) KMT2AMEN1POLBL3MBTL1ALDH1A1
SCHEMBL7639037 0.69 MEN1 (0.39) KMT2AMEN1POLBL3MBTL1ALDH1A1
SCHEMBL5207266 0.69 GSK3B (0.46) POLBGPR35TDP1L3MBTL1GSK3B
SCHEMBL2497335 0.68 POLB (0.39) KMT2AMEN1POLBTDP1
SCHEMBL2493216 0.68 POLB (0.44) KMT2AMEN1POLBTDP1ALDH1A1
SCHEMBL2494264 0.66 POLB (0.41) KMT2AMEN1POLB
SCHEMBL3836429 0.66 POLB (0.55) KMT2APOLBGPR35TDP1L3MBTL1
SCHEMBL2808786 0.64 GSK3B (0.50) KMT2AMEN1POLBGPR35TDP1
Hydrochloric Acid SCHEMBL7810688 0.64 POLB (0.53) KMT2APOLBGPR35TDP1L3MBTL1
SCHEMBL27363412 0.64 GPR35 (0.46) KMT2APOLBGPR35TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0970036-A1 ARYL- AND HETEROARYLCYCLOHEXENYL SUBSTITUTED ALKENES HAVING RETINOID AGONIST, ANTAGONIST OR INVERSE AGONIST TYPE BIOLOGICAL ACTIVITY Allergan Sales, Inc. (US) 2000-01-12 EP disclosed
WO-1998039284-A1 ARYL- AND HETEROARYLCYCLOHEXENYL SUBSTITUTED ALKENES HAVING RETINOID AGONIST, ANTAGONIST OR INVERSE AGONIST TYPE BIOLOGICAL ACTIVITY ALLERGAN SALES, INC. (US) 1998-09-11 WO disclosed