SCHEMBL8189802

SCHEMBL8189802

CCCCC(CO)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)NS(=O)(=O)c1cccc2c(N(C)C)cccc12

nearest known ligand 0.51

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
GLB1 P16278 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8773040 0.87 GLB1 (0.43) GLB1
SCHEMBL7378486 0.80 ALDH1A1 (0.44)
SCHEMBL1168296 0.78
SCHEMBL10963011 0.78
SCHEMBL29632046 0.78
SCHEMBL1168294 0.78
SCHEMBL7066334 0.78 TYMS (0.52) GLB1
SCHEMBL3813102 0.78 TYMS (0.52) GLB1
SCHEMBL6805481 0.78 TYMS (0.52) GLB1
SCHEMBL7333226 0.74 PLAU (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5872101-A Methods of treating neurodegenerative disorders using protease inhibitors SIBIA NEUROSCIENCES, INC. (US) 1999-02-16 US claimed
US-5863902-A Methods of treating neurodegenerative disorders using protease inhibitors SIBIA NEUROSCIENCES, INC. (US) 1999-01-26 US claimed
WO-1996020725-A2 PEPTIDE, PEPTIDE ANALOG AND AMINO ACID ANALOG PROTEASE INHIBITORS SIBIA NEUROSCIENCES, INC. (US) 1996-07-11 WO claimed
US-6017887-A Peptide, peptide analog and amino acid analog protease inhibitors SIBIA NEUROSCIENCES, INC. (US) 2000-01-25 US disclosed
US-5969100-A Peptide, peptide analog and amino acid analog protease inhibitors SIBIA NEUROSCIENCES, INC. (US) 1999-10-19 US disclosed
US-5872101-A Methods of treating neurodegenerative disorders using protease inhibitors SIBIA NEUROSCIENCES, INC. (US) 1999-02-16 US disclosed
US-5863902-A Methods of treating neurodegenerative disorders using protease inhibitors SIBIA NEUROSCIENCES, INC. (US) 1999-01-26 US disclosed
WO-1996020725-A2 PEPTIDE, PEPTIDE ANALOG AND AMINO ACID ANALOG PROTEASE INHIBITORS SIBIA NEUROSCIENCES, INC. (US) 1996-07-11 WO disclosed