SCHEMBL8190396

SCHEMBL8190396

Brc1ccc2[nH]c(-c3ccc[nH]3)nc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.48
PDPK1 O15530 1/20 0.45
IDO1 P14902 1/20 0.43
MMP13 P45452 4/20 0.40
NPC1 O15118 3/20 0.40
MMP2 P08253 3/20 0.40
MMP9 P14780 3/20 0.40
MMP8 P22894 3/20 0.40
GBA1 P04062 1/20 0.40
ATM Q13315 2/20 0.40
RAB9A P51151 2/20 0.40
ERAP1 Q9NZ08 1/20 0.40
AHR P35869 2/20 0.40
CYP2A6 P11509 1/20 0.40
NR4A2 P43354 1/20 0.40
RXFP1 Q9HBX9 1/20 0.38
PTGES O14684 2/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ABCB11 O95342 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8190402 0.88 ESR1 (0.62) ESR1PDPK1MMP13MMP2MMP9
SCHEMBL6754599 0.82 ESR1 (0.50) ESR1PDPK1MMP13NPC1MMP2
SCHEMBL3195220 0.81 SMN1; SMN2 (0.45) NPC1GBA1ATMRAB9AERAP1
SCHEMBL2053008 0.81 AMY1A (0.41) NPC1GBA1ATMRAB9AERAP1
SCHEMBL1170673 0.81 PDPK1 (0.51) ESR1PDPK1MMP13NPC1MMP2
SCHEMBL2048080 0.78 NPC1 (0.64) NPC1GBA1RAB9AALDH1A1KDM4E
SCHEMBL4842275 0.76 CDK5 (0.37) ESR1IDO1NPC1ATMRAB9A
SCHEMBL3201183 0.76 NPBWR1 (0.51) MMP13NPC1MMP2MMP9MMP8
SCHEMBL6753170 0.76 F2 (0.56)
SCHEMBL3340103 0.76 ATM (0.63) PDPK1MMP13NPC1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156779-A FUNGICIDES AGAINST CANDIDA UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2000-12-05 US disclosed
EP-0831832-A1 METHODS OF COMBATTING INFECTIOUS DISEASES USING DICATIONIC BIS-BENZIMIDAZOLES THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1998-04-01 EP disclosed
WO-1996040997-A1 METHOD OF FLUORESCENT DETECTION OF NUCLEIC ACIDS AND CYTOSKELETON ELEMENTS USING BIS-DICATIONIC ARYL FURANS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1996-12-19 WO disclosed
WO-1996040145-A1 METHODS OF COMBATTING INFECTIOUS DISEASES USING DICATIONIC BIS-BENZIMIDAZOLES THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1996-12-19 WO disclosed