SCHEMBL8190895

SCHEMBL8190895

O=C(O)c1ccc(Cl)c(-n2cccc2)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.55
ALDH1A1 P00352 3/20 0.49
TDP1 Q9NUW8 2/20 0.49
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2C19 P33261 1/20 0.48
MAPT P10636 1/20 0.46
SRD5A2 P31213 1/20 0.44
TTR P02766 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA9 Q16790 1/20 0.42
KMO O15229 1/20 0.41
ALK Q9UM73 1/20 0.41
ALOX15 P16050 1/20 0.41
MYC P01106 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
SERPINE1 P05121 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27772892 0.86 TSHR (0.55) TSHRALDH1A1TDP1CYP1A2CYP3A4
SCHEMBL7815535 0.80 MYC (0.57) ALDH1A1TDP1CYP2C19MAPTTTR
SCHEMBL5533223 0.77 KMT2A (0.60) TSHRALDH1A1TDP1CYP1A2CYP2C19
SCHEMBL31213040 0.76 MYC (0.57) TSHRALDH1A1TDP1CYP2C19MAPT
SCHEMBL29171465 0.75 KDM4E (0.57) ALDH1A1TDP1MAPTALOX15MYC
SCHEMBL20945174 0.74 ALDH1A1 (0.58) TSHRALDH1A1TDP1MAPTSRD5A2
SCHEMBL14502327 0.73 TDP1 (0.56) TSHRALDH1A1TDP1CYP2C19MAPT
SCHEMBL13903445 0.72 TSHR (0.52) TSHRALDH1A1TDP1MAPTSRD5A2
SCHEMBL15122952 0.72 GAA (0.62) TSHRALDH1A1TDP1TTRKMO
SCHEMBL371998 0.72 TSHR (1.00) TSHRALDH1A1MAPTSRD5A2TTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6162918-A Xanthene and acridine derivatives HOFFMANN-LA ROCHE INC. (US) 2000-12-19 US disclosed
US-5969139-A INHIBITORS OF HERPES SIMPLEX VIRUS THYMIDINE KINASE HOFFMANN-LA ROCHE INC. (US) 1999-10-19 US disclosed
EP-0823426-A1 Xanthene and acridine derivatives and their use F. HOFFMANN-LA ROCHE AG (CH) 1998-02-11 EP disclosed