SCHEMBL8191990

SCHEMBL8191990

NC(=O)c1ccc(-n2[nH]cc(-c3cccnc3)c2=O)nc1

nearest known ligand 0.70

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
P4HTM Q9NXG6 11/20 0.70
EGLN1 Q9GZT9 3/20 0.70
VHL P40337 6/20 0.67
MKNK1 Q9BUB5 1/20 0.52
MKNK2 Q9HBH9 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3610000 0.99 P4HTM (0.69) P4HTMEGLN1VHLMKNK1MKNK2
SCHEMBL3599948 0.89 P4HTM (0.72) P4HTMEGLN1VHLMKNK1MKNK2
Hydrochloric Acid SCHEMBL3611236 0.88 P4HTM (0.70) P4HTMEGLN1VHL
SCHEMBL3617392 0.88 P4HTM (0.70) P4HTMEGLN1VHL
Hydrochloric Acid SCHEMBL3842101 0.83 P4HTM (0.66) P4HTMEGLN1VHL
SCHEMBL8182341 0.83 P4HTM (0.72) P4HTMEGLN1VHL
SCHEMBL8257164 0.83 P4HTM (0.66) P4HTMEGLN1VHL
SCHEMBL8191995 0.83 EGLN1 (1.00) P4HTMEGLN1VHL
SCHEMBL3591779 0.82 VHL (0.71) P4HTMEGLN1VHL
SCHEMBL8186022 0.82 VHL (0.71) P4HTMEGLN1VHL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2097404-B1 SUBSTITUTED DIPYRIDYL-DIHYDROPYRAZOLONES AND USE THEREOF BAYER IP GMBH (DE) 2016-07-27 EP disclosed
US-20100093803-A1 SUBSTITUTED DIPYRIDYL-DIHYDROPYRAZOLONES AND USE THEREOF BAYER SCHERRING PHARMA AKTIENGELLSCHAFT (DE) 2010-04-15 US disclosed
WO-2008067874-A1 SUBSTITUTED DIPYRIDYL-DIHYDROPYRAZOLONES AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-06-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100093803-A1 SUBSTITUTED DIPYRIDYL-DIHYDROPYRAZOLONES AND USE THEREOF DCK, THPO, QDPR P4HTM 412/4885EGLN1 882/4885VHL 25/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.