SCHEMBL8192076

SCHEMBL8192076

COc1ccc(COC[C@H]2O[C@@H](n3c4cc(F)c(F)cc4c4c5c(c6c7cc(F)c(F)cc7[nH]c6c43)C(=O)NC5=O)[C@H](OCc3ccccc3)[C@@H](OCc3ccccc3)[C@@H]2OCc2ccccc2)cc1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 14/20 0.52
CCNE2 O96020 3/20 0.38
CDK4 P11802 3/20 0.38
CCND1 P24385 3/20 0.38
CCNE1 P24864 3/20 0.38
CDK2 P24941 3/20 0.38
PRKACA P17612 1/20 0.38
PRKACG P22612 1/20 0.38
PRKACB P22694 1/20 0.38
HTR1A P08908 1/20 0.37
ROCK2 O75116 2/20 0.36
CAMK2B Q13554 1/20 0.36
CAMK2G Q13555 1/20 0.36
CAMK2D Q13557 1/20 0.36
CAMK2A Q9UQM7 1/20 0.36
BCHE P06276 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5870061 0.90 TOP1 (0.58) TOP1CCNE2CDK4CCND1CCNE1
SCHEMBL6724824 0.89 TOP1 (0.61) TOP1
SCHEMBL5870514 0.89 TOP1 (0.61) TOP1
SCHEMBL7861913 0.87 TOP1 (0.65) TOP1
SCHEMBL7861934 0.83 TOP1 (0.42) TOP1HTR1ABCHE
SCHEMBL7024637 0.83 TOP1 (0.51) TOP1CCNE2CDK4CCND1CCNE1
SCHEMBL7860461 0.83 TOP1 (0.54) TOP1CCNE2CDK4CCND1CCNE1
SCHEMBL5870062 0.82 TOP1 (0.54) TOP1CCNE2CDK4CCND1CCNE1
SCHEMBL5870241 0.80 TOP1 (0.51) TOP1CCNE2CDK4CCND1CCNE1
SCHEMBL6731989 0.79 TOP1 (0.62) TOP1CCNE2CDK4CCND1CCNE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0971717-A4 CYTOTOXIC AMINO SUGAR AND RELATED SUGAR DERIVATIVES OF INDOLOPYRROLOCARBAZOLES BRISTOL MYERS SQUIBB CO (US) 2000-04-12 EP disclosed
EP-0971717-A1 CYTOTOXIC AMINO SUGAR AND RELATED SUGAR DERIVATIVES OF INDOLOPYRROLOCARBAZOLES Bristol-Myers Squibb Company (US) 2000-01-19 EP disclosed
WO-1998007433-A1 CYTOTOXIC AMINO SUGAR AND RELATED SUGAR DERIVATIVES OF INDOLOPYRROLOCARBAZOLES BRISTOL-MYERS SQUIBB COMPANY (US) 1998-02-26 WO disclosed