SCHEMBL8192202

SCHEMBL8192202

OCc1cccnc1-c1cccnc1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.50
KCNA5 P22460 2/20 0.41
CCR9 P51686 1/20 0.41
S100A4 P26447 2/20 0.41
CDC25B P30305 1/20 0.41
DHODH Q02127 2/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
KDM4E B2RXH2 2/20 0.39
GAA P10253 2/20 0.39
LMNA P02545 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
HTT P42858 1/20 0.39
MAPK1 P28482 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
TDP2 O95551 1/20 0.38
NSD2 O96028 1/20 0.38
ABL1 P00519 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11632316 0.84 DPP4 (0.71) DPP4KCNA5CCR9S100A4CDC25B
SCHEMBL30850781 0.81
SCHEMBL580627 0.81
SCHEMBL7160604 0.80 KDM4E (0.48) DPP4KCNA5CCR9NPC1RAB9A
SCHEMBL30832971 0.80 KDM4E (0.48) DPP4KCNA5CCR9NPC1RAB9A
SCHEMBL27838509 0.79 DPP4 (0.42) DPP4KCNA5S100A4CDC25BDHODH
SCHEMBL11737373 0.77 DPP4 (0.45) DPP4KCNA5S100A4CDC25BNPC1
SCHEMBL4049174 0.76 TRPV1 (0.47) DPP4KCNA5CCR9NPC1RAB9A
Alcohol SCHEMBL28672975 0.76 KDM4E (0.44) NPC1RAB9AKDM4EGAALMNA
SCHEMBL3431234 0.75 ALDH1A1 (0.48) DPP4S100A4CDC25BDHODHGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6136810-A DRUGS AS ENZYME INHIBITORS OF PHOSPHODIESTERASE YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-0885894-A1 PYRIDO [2,3-D] PYRIMIDINE DERIVATIVES AND MEDICINAL COMPOSITIONS THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1998-12-23 EP disclosed