SCHEMBL8192550

SCHEMBL8192550

O=C(CC1CCc2cc(OCc3ccccc3)ccc2C1=O)N[C@@H](Cc1ccccc1)C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.56
ITGA2B P08514 1/20 0.56
YAP1 P46937 5/20 0.52
GPR34 Q9UPC5 8/20 0.50
GPR132 Q9UNW8 2/20 0.50
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
PPARG P37231 1/20 0.46
CYP26A1 O43174 1/20 0.45
CYP24A1 Q07973 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8199673 0.93 ITGB3 (0.57) ITGB3ITGA2BYAP1GPR34GPR132
SCHEMBL8199071 0.93 ITGB3 (0.59) ITGB3ITGA2BYAP1GPR34GPR132
SCHEMBL8198563 0.91 ITGB3 (0.54) ITGB3ITGA2BYAP1MAOAMAOB
SCHEMBL8200056 0.87 ITGB3 (0.54) ITGB3ITGA2BGPR132MAOAMAOB
SCHEMBL8198782 0.86 ITGB3 (0.55) ITGB3ITGA2BMAOAMAOBCYP26A1
SCHEMBL8198784 0.86 ITGB3 (0.55) ITGB3ITGA2BMAOAMAOBCYP26A1
SCHEMBL8200699 0.86 ITGB3 (0.55) ITGB3ITGA2BMAOAMAOBCYP26A1
SCHEMBL8200304 0.84 ITGB3 (0.60) ITGB3ITGA2BMAOAMAOBCYP26A1
SCHEMBL8203736 0.82 ITGB3 (0.57) ITGB3ITGA2BMAOAMAOBCYP26A1
SCHEMBL8200229 0.80 ITGB3 (0.54) ITGB3ITGA2BMAOAMAOBCYP26A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed