SCHEMBL8203736

SCHEMBL8203736

O=C(CC1CCc2cc(OCc3ccccc3)ccc2C1=O)NC1Cc2ccccc2C1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.57
ITGA2B P08514 1/20 0.57
MAOA P21397 3/20 0.47
MAOB P27338 3/20 0.47
TAOK1 Q7L7X3 1/20 0.47
TAOK3 Q9H2K8 1/20 0.47
CYP24A1 Q07973 4/20 0.45
CYP26A1 O43174 3/20 0.45
FAAH O00519 7/20 0.44
CYP27A1 Q02318 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
DGAT1 O75907 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8200304 0.85 ITGB3 (0.60) ITGB3ITGA2BMAOAMAOBCYP24A1
SCHEMBL8199673 0.83 ITGB3 (0.57) ITGB3ITGA2BMAOAMAOBCYP24A1
SCHEMBL8192550 0.82 ITGB3 (0.56) ITGB3ITGA2BMAOAMAOBCYP24A1
SCHEMBL8198782 0.81 ITGB3 (0.55) ITGB3ITGA2BMAOAMAOBCYP24A1
SCHEMBL8198784 0.81 ITGB3 (0.55) ITGB3ITGA2BMAOAMAOBCYP24A1
SCHEMBL8200699 0.81 ITGB3 (0.55) ITGB3ITGA2BMAOAMAOBCYP24A1
SCHEMBL8200229 0.80 ITGB3 (0.54) ITGB3ITGA2BMAOAMAOBCYP24A1
SCHEMBL8198563 0.80 ITGB3 (0.54) ITGB3ITGA2BMAOAMAOBCYP24A1
SCHEMBL8199071 0.80 ITGB3 (0.59) ITGB3ITGA2BMAOAMAOBCYP24A1
SCHEMBL8200056 0.80 ITGB3 (0.54) ITGB3ITGA2BMAOAMAOBCYP24A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed