SCHEMBL8195082

SCHEMBL8195082

CCCC1CCc2sccc2C(N)=N1

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 17/20 0.49
NOS3 P29474 14/20 0.49
NOS1 P29475 10/20 0.49
DRD2 P14416 2/20 0.35
DRD3 P35462 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8193561 0.78 NOS2 (0.47) NOS2NOS3NOS1
SCHEMBL8194949 0.72 NOS2 (0.43) NOS2NOS3NOS1
SCHEMBL8063238 0.69 NOS2 (0.60) NOS2NOS3NOS1DRD2DRD3
SCHEMBL3842816 0.68 HTR2C (0.51) NOS2DRD2DRD3
Hydrochloric Acid SCHEMBL8100806 0.68 NOS2 (0.59) NOS2NOS3NOS1DRD2DRD3
SCHEMBL8193657 0.67 NOS2 (0.43) NOS2NOS3NOS1
SCHEMBL8193125 0.67 NOS2 (0.58) NOS2NOS3NOS1
SCHEMBL8060969 0.67 NOS2 (1.00) NOS2NOS3NOS1
SCHEMBL8214849 0.66 NOS3 (1.00) NOS2NOS3NOS1
Iodide SCHEMBL8099764 0.65 NOS2 (0.96) NOS2NOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000064904-A1 5,7-BICYCLIC AMIDINE DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS ASTRAZENECA AB (SE) 2000-11-02 WO claimed
WO-2000064904-A1 5,7-BICYCLIC AMIDINE DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS ASTRAZENECA AB (SE) 2000-11-02 WO disclosed