SCHEMBL8195802

SCHEMBL8195802

COc1cc(-c2c(C(F)(F)F)n[nH]c2-c2ccc(S(=O)(=O)CCCO)cc2)ccc1Br

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 3/20 0.37
NR1H3 Q13133 3/20 0.37
FYN P06241 1/20 0.36
AURKA O14965 1/20 0.36
NTRK1 P04629 1/20 0.36
KDR P35968 1/20 0.36
AURKB Q96GD4 1/20 0.36
CA2 P00918 2/20 0.36
ALDH1A1 P00352 1/20 0.34
PTGS2 P35354 1/20 0.34
TP53 P04637 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAPT P10636 2/20 0.34
LMNA P02545 1/20 0.34
HPGD P15428 1/20 0.34
KMT2A Q03164 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CHEK1 O14757 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8188363 0.94 FYN (0.38) FYNAURKANTRK1KDRAURKB
SCHEMBL8194835 0.87 PTGS2 (0.41) NR1H2NR1H3ALDH1A1PTGS2TP53
SCHEMBL8187629 0.84 PTGS2 (0.41) CA2ALDH1A1PTGS2TP53SMN1; SMN2
SCHEMBL8200043 0.84 PTGS2 (0.40) CA2ALDH1A1PTGS2TP53SMN1; SMN2
SCHEMBL8196703 0.81 PTGS2 (0.42) ALDH1A1PTGS2LMNAKMT2A
SCHEMBL8199177 0.79 PTGS2 (0.41) FYNAURKANTRK1KDRAURKB
SCHEMBL8196846 0.79 AR (0.39) AURKANTRK1KDRAURKBALDH1A1
SCHEMBL8201315 0.79 KDM4E (0.34) FYNALDH1A1PTGS2MAPTCHEK1
SCHEMBL8196932 0.78 HTT (0.41) PTGS2SMN1; SMN2MAPTKMT2ANPSR1
SCHEMBL8188386 0.78 NR1H2 (0.40) NR1H2NR1H3PTGS2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO claimed
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed