SCHEMBL8196846

SCHEMBL8196846

COc1ccc(-c2c(C(F)(F)F)n[nH]c2-c2ccc(S(=O)(=O)CCO)cc2)cc1C#N

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
AR P10275 3/20 0.39
AURKA O14965 1/20 0.36
NTRK1 P04629 1/20 0.36
KDR P35968 1/20 0.36
AURKB Q96GD4 1/20 0.36
F11 P03951 1/20 0.35
RORC P51449 1/20 0.34
ALDH1A1 P00352 2/20 0.34
PGR P06401 1/20 0.34
SCN9A Q15858 1/20 0.33
GPBAR1 Q8TDU6 1/20 0.33
CXCR2 P25025 1/20 0.33
SLC22A12 Q96S37 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8200042 0.87 AR (0.37) ARAURKANTRK1KDRAURKB
SCHEMBL8196703 0.86 PTGS2 (0.42) ALDH1A1
SCHEMBL8188363 0.84 FYN (0.38) AURKANTRK1KDRAURKBALDH1A1
SCHEMBL8196932 0.81 HTT (0.41)
SCHEMBL8188386 0.81 NR1H2 (0.40)
SCHEMBL8194835 0.81 PTGS2 (0.41) ALDH1A1
SCHEMBL8199177 0.80 PTGS2 (0.41) AURKANTRK1KDRAURKBALDH1A1
SCHEMBL8187629 0.80 PTGS2 (0.41) ALDH1A1
SCHEMBL8200043 0.79 PTGS2 (0.40) ALDH1A1
SCHEMBL8195802 0.79 NR1H2 (0.37) AURKANTRK1KDRAURKBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO claimed
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed