SCHEMBL8196643

SCHEMBL8196643

Cc1cc(-c2cc(-c3ccc(S(=O)(=O)CCCO)cc3)[nH]n2)ccc1F

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.40
PTGS1 P23219 2/20 0.39
CA2 P00918 5/20 0.39
CA1 P00915 1/20 0.38
CA5A P35218 1/20 0.38
CA5B Q9Y2D0 1/20 0.38
NPC1 O15118 2/20 0.36
MAPT P10636 2/20 0.36
RAB9A P51151 2/20 0.36
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36
PKM P14618 1/20 0.36
KMT2A Q03164 1/20 0.36
MCL1 Q07820 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PHGDH O43175 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8196087 0.93 PTGS2 (0.41) PTGS2PTGS1CA2CA1CA5A
SCHEMBL8202086 0.87 RAF1 (0.41) PTGS2PTGS1CA2NPC1MAPT
SCHEMBL8188094 0.85 MEN1 (0.45) CA2NPC1RAB9AMEN1POLB
SCHEMBL8196192 0.85 CA2 (0.39) PTGS2PTGS1CA2NPC1MAPT
SCHEMBL8202081 0.83 KMT2A (0.53) CA2NPC1MAPTRAB9AMEN1
SCHEMBL8195997 0.81 BCHE (0.43) CA2NPC1MAPTRAB9AMEN1
SCHEMBL8201936 0.80 RAF1 (0.42) PTGS2PTGS1CA2NPC1MAPT
SCHEMBL8195766 0.79 CA2 (0.40) CA2NPC1MAPTRAB9AMEN1
SCHEMBL8196977 0.78 APP (0.41) CA2NPC1MAPTRAB9AMEN1
SCHEMBL8188503 0.78 PTGS2 (0.40) PTGS2PTGS1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO claimed
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed