SCHEMBL8198380

SCHEMBL8198380

CC(NC(=O)C(Cc1c[nH]c2ccc(F)cc12)NC(=O)O)c1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 2/20 0.63
MMP8 P22894 2/20 0.63
MMP2 P08253 1/20 0.55
TACR1 P25103 2/20 0.53
ITGB2 P05107 2/20 0.50
ICAM1 P05362 2/20 0.50
ITGAL P20701 2/20 0.50
HTR2A P28223 1/20 0.50
HTR2C P28335 1/20 0.50
TSHR P16473 1/20 0.48
ACE P12821 1/20 0.47
ECE1 P42892 5/20 0.47
TGM2 P21980 1/20 0.46
NR3C1 P04150 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8198377 1.00 MMP9 (0.63) MMP9MMP8MMP2TACR1ITGB2
SCHEMBL8850370 0.87 MMP9 (0.80) MMP9MMP8MMP2TACR1ACE
SCHEMBL8201151 0.87 MMP9 (0.80) MMP9MMP8MMP2TACR1ACE
SCHEMBL8201153 0.87 MMP9 (0.80) MMP9MMP8MMP2TACR1ACE
SCHEMBL8488113 0.84 MMP9 (0.51) MMP9MMP8MMP2TACR1ITGB2
SCHEMBL8487186 0.83 HTR2A (0.50) MMP9MMP8MMP2TACR1ITGB2
SCHEMBL21292855 0.80 HTR2A (0.61) HTR2AHTR2CTSHRNR3C1
SCHEMBL20425196 0.80 HTR2A (0.61) HTR2AHTR2CTSHRNR3C1
SCHEMBL20242715 0.80 HTR2A (0.61) HTR2AHTR2CTSHRNR3C1
SCHEMBL8481429 0.78 MMP9 (0.76) MMP9MMP8MMP2TACR1ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000930-A2 Tachykinin antagonists WARNER-LAMBERT COMPANY (US) 2000-05-17 EP claimed
EP-0655055-A1 TACHYKININ ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1995-05-31 EP claimed
WO-1994004494-A1 TACHYKININ ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1994-03-03 WO claimed
EP-1000930-A2 Tachykinin antagonists WARNER-LAMBERT COMPANY (US) 2000-05-17 EP disclosed
US-5981755-A Tachykinin antagonists WARNER-LAMBERT COMPANY (US) 1999-11-09 US disclosed
US-5594022-A CARBAMATES WARNER-LAMBERT COMPANY (US) 1997-01-14 US disclosed
WO-1994004494-A1 TACHYKININ ANTAGONISTS WARNER-LAMBERT COMPANY (US) 1994-03-03 WO disclosed