SCHEMBL8487186

SCHEMBL8487186

CC(NC(=O)C(Cc1c[nH]c2ccc(F)cc12)OC(N)=O)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.50
MMP9 P14780 2/20 0.50
MMP8 P22894 2/20 0.50
HTR2C P28335 1/20 0.50
TACR1 P25103 3/20 0.46
NOTUM Q6P988 2/20 0.46
MPO P05164 3/20 0.46
TSHR P16473 1/20 0.46
SLC6A4 P31645 1/20 0.45
MMP2 P08253 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43
ITGB2 P05107 1/20 0.43
ICAM1 P05362 1/20 0.43
ITGAL P20701 1/20 0.43
SOS1 Q07889 1/20 0.43
SCN9A Q15858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8483346 0.88 MMP9 (0.63) MMP9MMP8TACR1MMP2MEN1
SCHEMBL8198380 0.83 MMP9 (0.63) HTR2AMMP9MMP8HTR2CTACR1
SCHEMBL8198377 0.83 MMP9 (0.63) HTR2AMMP9MMP8HTR2CTACR1
SCHEMBL28822903 0.79 HTR2A (0.64) HTR2AHTR2CNOTUMMPOTSHR
SCHEMBL28504603 0.79 HTR2A (0.64) HTR2AHTR2CNOTUMMPOTSHR
SCHEMBL28504602 0.79 HTR2A (0.64) HTR2AHTR2CNOTUMMPOTSHR
SCHEMBL8481416 0.77 MMP9 (0.62) MMP9MMP8TACR1MMP2MEN1
SCHEMBL8850751 0.73 MMP9 (0.60) MMP9MMP8TACR1MMP2MEN1
SCHEMBL8850747 0.73 MMP9 (0.60) MMP9MMP8TACR1MMP2MEN1
SCHEMBL21292855 0.73 HTR2A (0.61) HTR2AHTR2CNOTUMMPOTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5856354-A RESPIRATORY SYSTEM DISORDERS, ANTIINFLAMMATORY AGENTS, GASTROINTESTINAL DISORDERS, VISION DEFECTS, ANTIALLERGENS,PAIN, NERVOUS SYSTEM DISORDERS, HEADACHES WARNER-LAMBERT COMPANY (US) 1999-01-05 US disclosed
US-5716979-A NONPEPTIDES, UNIQUE IN ALKYLATION/SUBSTITUTION PATTERN ALONG THEIR BACKBONE, USEFUL FOR TREATING DISORDERS SUCH AS RESPIRATORY, INFLAMMATORY, GASTROINTESTINAL, OPHTHALMIC, ALLERGIES, PAIN, VASCULAR, MIGRANE, ARTHRITIS AND BRAIN WARNER-LAMBERT COMPANY (US) 1998-02-10 US disclosed