SCHEMBL8198639

SCHEMBL8198639

C=C(O)c1nc(=O)[nH]c2ccccc12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 4/20 0.61
KDM4E B2RXH2 9/20 0.56
ALDH1A1 P00352 7/20 0.56
HSD17B10 Q99714 5/20 0.56
HPGD P15428 4/20 0.56
TSHR P16473 1/20 0.56
APP P05067 2/20 0.48
LMNA P02545 2/20 0.42
GLA P06280 2/20 0.42
GAA P10253 2/20 0.42
HTT P42858 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
ATM Q13315 1/20 0.42
DYRK1A Q13627 1/20 0.42
TDP1 Q9NUW8 1/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
CASP1 P29466 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MAPT P10636 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14072437 0.84 ADORA3 (0.68) ADORA3KDM4EALDH1A1HSD17B10HPGD
SCHEMBL29033598 0.80 ADORA3 (0.62) ADORA3KDM4EALDH1A1HSD17B10HPGD
SCHEMBL17753303 0.79 ADORA3 (0.61) ADORA3KDM4EALDH1A1HSD17B10HPGD
SCHEMBL17753301 0.79 ADORA3 (0.61) ADORA3KDM4EALDH1A1HSD17B10HPGD
SCHEMBL13995844 0.79 ADORA3 (0.61) ADORA3KDM4EALDH1A1HSD17B10HPGD
SCHEMBL30725575 0.79 ADORA3 (0.57) ADORA3KDM4EALDH1A1HSD17B10HPGD
SCHEMBL11487364 0.77 ADORA3 (0.58) ADORA3KDM4EALDH1A1HSD17B10HPGD
SCHEMBL31060760 0.76 ADORA3 (1.00) ADORA3KDM4EALDH1A1HSD17B10HPGD
SCHEMBL7417909 0.76 ADORA3 (0.57) ADORA3KDM4EALDH1A1HSD17B10HPGD
SCHEMBL554709 0.74 KDM4E (0.58) ADORA3KDM4EALDH1A1HSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008109180-A2 METALLOPROTEASE INHIBITORS CONTAINING A HETEROCYCLIC MOIETY ALANTOS PHARMACEUTICALS HOLDING, INC. (US) 2008-09-12 WO disclosed