SCHEMBL8199562

SCHEMBL8199562

O=C1[N]C(=O)c2cc([N+](=O)[O-])c(Cl)cc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.46
TSHR P16473 1/20 0.46
ALDH1A1 P00352 3/20 0.44
CYP3A4 P08684 2/20 0.44
VCAM1 P19320 5/20 0.41
PGK1 P00558 1/20 0.41
CA12 O43570 2/20 0.40
CA9 Q16790 2/20 0.40
DHFR P00374 1/20 0.40
MAPT P10636 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
LMNA P02545 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
STAT6 P42226 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3980207 0.77 TSHR (0.54) MAPK1TSHRALDH1A1CYP3A4VCAM1
SCHEMBL438752 0.77 CYP3A4 (0.50) MAPK1TSHRALDH1A1CYP3A4VCAM1
SCHEMBL11657285 0.77 ALDH1A1 (0.50) MAPK1TSHRALDH1A1CYP3A4VCAM1
SCHEMBL29835178 0.77 CYP3A4 (0.50) MAPK1TSHRALDH1A1CYP3A4VCAM1
SCHEMBL786237 0.77 CYP3A4 (0.50) MAPK1TSHRALDH1A1CYP3A4VCAM1
SCHEMBL1413188 0.76 AHR (0.45) MAPK1TSHRALDH1A1CA12CA9
SCHEMBL9180125 0.76 TSHR (0.62) MAPK1TSHRALDH1A1CYP3A4VCAM1
SCHEMBL28012095 0.76 CYP3A4 (0.49) MAPK1TSHRALDH1A1CYP3A4VCAM1
SCHEMBL441605 0.74 CA12 (0.47) MAPK1TSHRALDH1A1CYP3A4VCAM1
SCHEMBL5608736 0.74 TSHR (0.40) MAPK1TSHRALDH1A1CYP3A4VCAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6166082-A Substituted 5-biarylpentanoic acids and derivatives as matrix metalloprotease inhibitors BAYER CORPORATION (US) 2000-12-26 US disclosed