SCHEMBL5608736

SCHEMBL5608736

O=C1[N]Nc2cc(Cl)c([N+](=O)[O-])cc21

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
AKR1B1 P15121 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP3A4 P08684 1/20 0.39
VCAM1 P19320 5/20 0.38
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38
PKM P14618 1/20 0.37
PGK1 P00558 1/20 0.36
PDE7A Q13946 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5608587 0.76 SNCA (0.39) TSHRMAPK1ALDH1A1CYP3A4LMNA
SCHEMBL8199562 0.74 MAPK1 (0.46) TSHRMAPK1ALDH1A1CYP3A4VCAM1
SCHEMBL5608778 0.74 ALOX15 (0.41) MAPK1ALDH1A1CYP3A4
SCHEMBL8872707 0.72 CES1 (0.62) TSHRMAPK1AKR1B1ALDH1A1CYP3A4
SCHEMBL5608922 0.72 MAOA (0.40) MAPK1ALDH1A1CYP3A4
SCHEMBL29835178 0.70 CYP3A4 (0.50) TSHRMAPK1AKR1B1ALDH1A1CYP3A4
SCHEMBL438752 0.70 CYP3A4 (0.50) TSHRMAPK1AKR1B1ALDH1A1CYP3A4
SCHEMBL786237 0.70 CYP3A4 (0.50) TSHRMAPK1AKR1B1ALDH1A1CYP3A4
SCHEMBL5608967 0.70 SNCA (0.39) ALDH1A1LMNA
SCHEMBL6820729 0.70 PTPRC (0.50) ALDH1A1CYP3A4CA12CA9LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1797042-A1 INDOZOLONE DERIVATIVES AS 11B-HSD1 INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2007-06-20 EP disclosed
WO-2006034804-A1 INDOZOLONE DERIVATIVES AS 11B-HSD1 INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2006-04-06 WO disclosed