SCHEMBL8199717

SCHEMBL8199717

COc1ccc2c(c1)CC[C@@H](CN1CCC(c3ccccc3)CC1)[C@H]2O

nearest known ligand 0.67

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 1/20 0.53
CCR5 P51681 1/20 0.52
SLC18A3 Q16572 2/20 0.48
DRD2 P14416 1/20 0.46
SIGMAR1 Q99720 2/20 0.46
HTR1A P08908 1/20 0.46
GRIN1 Q05586 1/20 0.45
GRIN2B Q13224 1/20 0.45
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6490328 1.00 SLC6A9 (0.53) SLC6A9CCR5SLC18A3DRD2SIGMAR1
SCHEMBL8199718 1.00 SLC6A9 (0.53) SLC6A9CCR5SLC18A3DRD2SIGMAR1
SCHEMBL8236868 0.90 SLC6A9 (0.51) SLC6A9DRD2GRIN1GRIN2B
SCHEMBL5904205 0.85 SLC6A9 (0.46) SLC6A9SIGMAR1
SCHEMBL11525123 0.82 MAPT (0.46) SLC6A9
SCHEMBL6500564 0.82 CD274 (0.47) CCR5SLC18A3GRIN1GRIN2B
SCHEMBL8203174 0.79 HRH3 (0.45) SLC18A3DRD2SIGMAR1GRIN1GRIN2B
SCHEMBL8203170 0.79 HRH3 (0.45) SLC18A3DRD2SIGMAR1GRIN1GRIN2B
SCHEMBL8203171 0.79 HRH3 (0.45) SLC18A3DRD2SIGMAR1GRIN1GRIN2B
Hydrochloric Acid SCHEMBL9520222 0.78 ADRA2A (0.46) DRD2SIGMAR1HTR1ACA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed