SCHEMBL8200233

SCHEMBL8200233

N#CN(Cc1ccc(C(N)=O)cc1)C(N)=Nc1ccncc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.45
PLG P00747 1/20 0.37
NOS1 P29475 4/20 0.37
NOS3 P29474 3/20 0.34
NOS2 P35228 3/20 0.34
PLA2G10 O15496 1/20 0.34
PLA2G2A P14555 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
HIF1A Q16665 1/20 0.34
ABHD6 Q9BV23 1/20 0.34
IKBKE Q14164 1/20 0.34
TBK1 Q9UHD2 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
MYC P01106 1/20 0.33
PARP10 Q53GL7 1/20 0.33
HGFAC Q04756 1/20 0.32
KDM1A O60341 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8200238 0.86 PLG (0.40) CYP17A1PLGNOS1NOS3NOS2
SCHEMBL8218500 0.81 CYP17A1 (0.36) CYP17A1PLGNOS1NOS3NOS2
SCHEMBL7978140 0.76 CYP17A1 (0.43) CYP17A1PLGIKBKETBK1NPC1
SCHEMBL8195014 0.74 HTT (0.54) ALDH1A1CYP1A2CYP2D6
SCHEMBL504667 0.74 PLG (0.44) PLGNOS1NOS3NOS2
SCHEMBL504588 0.74 PLG (0.44) PLGNOS1NOS3NOS2
SCHEMBL7966282 0.73 GAA (0.43) ALDH1A1RAB9A
SCHEMBL9299302 0.72 PLG (0.42) PLGNOS1NOS3NOS2
SCHEMBL504564 0.71 PLG (0.41) PLGNOS1NOS3NOS2
SCHEMBL8200235 0.71 CYP17A1 (0.46) CYP17A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000061561-A1 CYANOGUANIDINE COMPOUNDS SHIONOGI BIORESEARCH CORP. (US) 2000-10-19 WO claimed
WO-2000061559-A1 N-SUBSTITUTED CYANOGUANIDINE COMPOUNDS SHIONOGI BIORESEARCH CORP. (US) 2000-10-19 WO disclosed