SCHEMBL8200380

SCHEMBL8200380

FC(F)(F)c1cccc(-c2ccccc2C2=NCCN2)c1

nearest known ligand 0.63

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 13/20 0.63
PTAFR P25105 1/20 0.47
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
MCL1 Q07820 1/20 0.46
PARP1 P09874 1/20 0.44
MAOB P27338 1/20 0.43
PARP10 Q53GL7 1/20 0.43
PARP11 Q9NR21 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8201787 0.89 NISCH (0.62) NISCH
SCHEMBL8189633 0.84 NISCH (0.71) NISCHALDH1A1
Hydrochloric Acid SCHEMBL8201249 0.83 NISCH (0.44) NISCHPTAFRALDH1A1PARP1MAOB
SCHEMBL8204316 0.81 NISCH (0.74) NISCHMAOB
SCHEMBL8202555 0.81 NISCH (0.48) NISCHPTAFRALDH1A1MAOBPARP10
SCHEMBL10822807 0.79 MAPT (0.52) NISCHALDH1A1LMNA
Hydrochloric Acid SCHEMBL7736305 0.79 NISCH (0.48) NISCHALDH1A1PARP1MAOB
SCHEMBL8201474 0.78 NISCH (0.69) NISCHMAOB
SCHEMBL17840165 0.78 RORC (0.57) ALDH1A1MAOB
Hydrochloric Acid SCHEMBL7736307 0.78 NISCH (0.42) NISCHALDH1A1PARP1MAOBPARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000078726-A1 IMIDAZOLINE DERIVATIVES FOR THE TREATMENT OF DIABETES, ESPECIALLY TYPE II DIABETES ELI LILLY AND COMPANY (US) 2000-12-28 WO disclosed