SCHEMBL8200721

SCHEMBL8200721

O=C(O)NCc1cccc(-c2ccc3c(c2)NC(=O)CO3)c1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.59
TSHR P16473 1/20 0.53
TP53 P04637 4/20 0.52
LMNA P02545 2/20 0.52
MAOA P21397 1/20 0.51
KMT2A Q03164 2/20 0.50
MAPT P10636 3/20 0.49
ALDH1A1 P00352 3/20 0.48
MAPK1 P28482 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
MMP12 P39900 1/20 0.47
MMP8 P22894 1/20 0.46
MMP13 P45452 1/20 0.46
NR3C2 P08235 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13343865 0.84 BRD4 (0.57) PARP1TSHRTP53LMNAMAOA
SCHEMBL4933671 0.81 MMP13 (0.58) PARP1MMP12MMP8MMP13
SCHEMBL4934583 0.81 PARP1 (0.53) PARP1KMT2AMAPTALDH1A1MAPK1
SCHEMBL304764 0.79 MAPT (0.62) PARP1LMNAKMT2AMAPTALDH1A1
SCHEMBL14073051 0.78 PARP1 (0.70) PARP1TSHRTP53LMNAMAOA
SCHEMBL27663635 0.78 PARP1 (0.45) PARP1TSHRTP53LMNAMAOA
SCHEMBL14073116 0.77 PARP1 (0.62) PARP1TSHRTP53LMNAMAOA
SCHEMBL4259329 0.77 PARP1 (0.65) PARP1KMT2AMAPTALDH1A1MAPK1
SCHEMBL531798 0.77 TSHR (0.74) PARP1TSHRTP53LMNAMAOA
SCHEMBL4267366 0.76 MMP12 (0.70) PARP1KMT2AMAPTALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008063668-A1 HETEROBICYCLIC METALLOPROTEASE INHIBITORS ALANTOS PHARMACEUTICALS HOLDING, INC. (US) 2008-05-29 WO disclosed