SCHEMBL8201028

SCHEMBL8201028

O=C1c2ccc(OCc3ccccc3-c3ccccc3)cc2CCC1C(=O)N1CCC(c2ccccc2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 2/20 0.45
CD274 Q9NZQ7 4/20 0.44
FFAR1 O14842 2/20 0.40
FFAR4 Q5NUL3 2/20 0.40
ADAM17 P78536 1/20 0.40
CCR5 P51681 1/20 0.39
ADRA1D P25100 1/20 0.39
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
MAPT P10636 3/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP24A1 Q07973 3/20 0.38
ALDH1A1 P00352 2/20 0.38
GAA P10253 2/20 0.38
CYP27A1 Q02318 2/20 0.38
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8200671 0.88 GRIN1 (0.48) ADRA1DADRA1AADRA1BRAB9ASMN1; SMN2
SCHEMBL8199368 0.81 CYP26A1 (0.49) CYP26A1CD274ADRA1DADRA1AADRA1B
SCHEMBL7130448 0.76 HRH3 (0.51) CD274ADRA1DADRA1AADRA1BITGB3
SCHEMBL8200806 0.75 CYP26A1 (0.45) CYP26A1CD274FFAR1FFAR4ADAM17
SCHEMBL8192688 0.75 CYP26A1 (0.45) CYP26A1CD274FFAR1FFAR4ADAM17
SCHEMBL8192685 0.75 CYP26A1 (0.45) CYP26A1CD274FFAR1FFAR4ADAM17
SCHEMBL6500564 0.74 CD274 (0.47) CD274CCR5ADRA1DADRA1AADRA1B
SCHEMBL8200598 0.72 CYP26A1 (0.52) CYP26A1CD274CYP24A1CYP27A1
SCHEMBL8202807 0.71 ADRA1D (0.46) CD274ADRA1DADRA1AADRA1BGRIN1
SCHEMBL8202799 0.71 ADRA1D (0.46) CD274ADRA1DADRA1AADRA1BGRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed